SCHEMBL14546705

SCHEMBL14546705

N#Cc1ccnc(CI)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 1/20 0.40
CLK4 Q9HAZ1 2/20 0.39
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
KCNH2 Q12809 1/20 0.35
NPY5R Q15761 1/20 0.35
LMNA P02545 2/20 0.33
VNN1 O95497 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
GRM5 P41594 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
CYP2A6 P11509 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
CDC7 O00311 4/20 0.32
CDK2 P24941 2/20 0.32
MAP3K14 Q99558 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7666624 0.84 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8KCNH2
SCHEMBL3242600 0.80 CYP1A2 (0.44) MBOAT4CLK4CCNCCDK8KCNH2
SCHEMBL16532586 0.80 MBOAT4 (0.43) MBOAT4CLK4CCNCCDK8LMNA
SCHEMBL3356564 0.80 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8KCNH2
SCHEMBL29478779 0.80 NOTUM (0.43) MBOAT4CLK4CCNCCDK8KCNH2
SCHEMBL30607265 0.80 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8LMNA
SCHEMBL17168474 0.80 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8KCNH2
SCHEMBL481078 0.80 NOTUM (0.43) MBOAT4CLK4CCNCCDK8KCNH2
SCHEMBL18078827 0.80 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8LMNA
Hydrochloric Acid SCHEMBL16517183 0.78 MBOAT4 (0.42) MBOAT4CLK4CCNCCDK8LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007048070-A2 PYRROLO-PYRIDINE DERIVATIVES FOR THE TREATMENT OF CANCER DISEASES AMGEN INC. (US) 2007-04-26 WO disclosed