SCHEMBL17168474

SCHEMBL17168474

N#Cc1ccnc(CF)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 1/20 0.40
CLK4 Q9HAZ1 1/20 0.39
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
NPY5R Q15761 6/20 0.35
KCNH2 Q12809 5/20 0.35
EGLN2 Q96KS0 1/20 0.34
VNN1 O95497 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
GRM5 P41594 1/20 0.33
KDM4C Q9H3R0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3356564 0.80 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8NPY5R
SCHEMBL3242600 0.80 CYP1A2 (0.44) MBOAT4CLK4CCNCCDK8NPY5R
SCHEMBL30607265 0.80 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8EGLN2
SCHEMBL14546705 0.80 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8NPY5R
SCHEMBL7666624 0.80 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8NPY5R
SCHEMBL29478779 0.80 NOTUM (0.43) MBOAT4CLK4CCNCCDK8NPY5R
SCHEMBL16532586 0.80 MBOAT4 (0.43) MBOAT4CLK4CCNCCDK8VNN1
SCHEMBL481078 0.80 NOTUM (0.43) MBOAT4CLK4CCNCCDK8NPY5R
SCHEMBL18078827 0.80 MBOAT4 (0.40) MBOAT4CLK4CCNCCDK8EGLN2
Hydrochloric Acid SCHEMBL16517183 0.78 MBOAT4 (0.42) MBOAT4CLK4CCNCCDK8VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9481650-B2 Process for the preparation of 2-trifluoromethyl isonicotinic acid and esters HOFFMANN LA ROCHE INC. (US) 2016-11-01 US disclosed
US-20150291530-A1 PROCESS FOR THE PREPARATION OF 2-TRIFLUOROMETHYL ISONICOTINIC ACID AND ESTERS HOFFMANN-LA ROCHE INC. (US) 2015-10-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150291530-A1 PROCESS FOR THE PREPARATION OF 2-TRIFLUOROMETHYL ISONICOTINIC ACID AND ESTERS TAAR1, TAAR5, TSHR MBOAT4 999/4885CLK4 4674/4885CCNC 3721/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.