SCHEMBL14548784

SCHEMBL14548784

COC(=O)c1cc(I)cnc1CI

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 13/20 0.44
TSHR P16473 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA7 P43166 2/20 0.34
CA9 Q16790 2/20 0.34
CA14 Q9ULX7 2/20 0.34
PDK2 Q15119 1/20 0.34
PDK4 Q16654 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL215798 0.78 OPRK1 (0.47) OPRK1TSHRKDM4EALDH1A1GLA
SCHEMBL8091281 0.78 OPRK1 (0.47) OPRK1TSHRKDM4EALDH1A1GLA
SCHEMBL1505507 0.77 OPRK1 (0.46) OPRK1TSHRKDM4EALDH1A1GLA
SCHEMBL2420694 0.77 OPRK1 (0.46) OPRK1TSHRKDM4EALDH1A1GLA
SCHEMBL6775808 0.76 OPRK1 (0.43) OPRK1KDM4EALDH1A1GLAGAA
SCHEMBL2436219 0.75 OPRK1 (0.45) OPRK1TSHRKDM4EALDH1A1GLA
SCHEMBL8274376 0.75 KDM4E (0.49) KDM4EALDH1A1GAA
SCHEMBL6713858 0.72 DPP4 (0.45) TSHRALDH1A1CA12CA1CA2
SCHEMBL20184058 0.69 OPRK1 (0.48) OPRK1
SCHEMBL21171175 0.69 OPRK1 (0.74) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8349872-B2 Tripyridyl carboxamide orexin receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-01-08 US disclosed