SCHEMBL14554188

SCHEMBL14554188

O=C(CO)Nc1cccc(-c2nn(C3CCCCO3)c3ccc(-c4ncn(C(c5ccccc5)(c5ccccc5)c5ccccc5)n4)cc23)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 4/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
FGFR1 P11362 1/20 0.34
DDR2 Q16832 1/20 0.34
MCL1 Q07820 1/20 0.34
DGAT2 Q96PD7 1/20 0.33
MAPT P10636 5/20 0.33
LMNA P02545 2/20 0.33
PIP5K1C O60331 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
IDH2 P48735 1/20 0.32
CPT2 P23786 1/20 0.31
CPT1A P50416 1/20 0.31
TP53 P04637 2/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5397809 0.93 PTPN1 (0.36) MAP4K4RXRARXRBRXRGFGFR1
SCHEMBL5386995 0.93 MAPT (0.38) MAP4K4RXRARXRBRXRGFGFR1
SCHEMBL5383426 0.92 MAP4K4 (0.38) MAP4K4FGFR1DDR2NPC1ALDH1A1
SCHEMBL5373247 0.92 ECE1 (0.38) MAP4K4RXRARXRBRXRGFGFR1
SCHEMBL5391965 0.92 FGFR1 (0.36) MAP4K4RXRARXRBRXRGFGFR1
SCHEMBL5380244 0.92 MMP2 (0.36) MAP4K4RXRARXRBRXRGFGFR1
SCHEMBL5380109 0.92 L3MBTL1 (0.39) MAP4K4RXRARXRBRXRGFGFR1
SCHEMBL5372575 0.92 MAP4K4 (0.38) MAP4K4RXRARXRBRXRGFGFR1
SCHEMBL5378724 0.91 SMN1; SMN2 (0.39) MAP4K4FGFR1DDR2MCL1MAPT
SCHEMBL5377561 0.90 FGFR1 (0.34) MAP4K4RXRARXRBRXRGFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130011923-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-01-10 US disclosed