SCHEMBL14558488

SCHEMBL14558488

CC(C)NCc1cccc(C(N)=O)c1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEP1B Q16820 11/20 0.54
KDM1A O60341 1/20 0.49
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
F10 P00742 1/20 0.49
PARP1 P09874 1/20 0.47
IDH1 O75874 1/20 0.47
VNN1 O95497 1/20 0.46
AURKA O14965 1/20 0.45
RPS6KB1 P23443 1/20 0.45
AURKB Q96GD4 1/20 0.45
FOLH1 Q04609 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19091172 0.86 MEP1B (0.53) MEP1BKDM1AMAOAMAOBF10
SCHEMBL17788675 0.85 MEP1B (0.71) MEP1BFOLH1
SCHEMBL6911637 0.85 MEP1B (0.55) MEP1BMAOB
SCHEMBL19954263 0.84 MEP1B (0.48) MEP1BKDM1AMAOAMAOBF10
SCHEMBL27119412 0.84 PRSS1 (0.57) MEP1BF10
SCHEMBL10331798 0.84 MEP1B (0.54) MEP1B
SCHEMBL19954186 0.84 MEP1B (0.48) MEP1BKDM1AMAOAMAOBF10
SCHEMBL5005534 0.84 MEP1B (0.52) MEP1BKDM1AMAOAMAOB
SCHEMBL23553939 0.83 ROCK2 (0.60) MEP1B
SCHEMBL19287247 0.83 MEP1B (0.52) MEP1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9914740-B2 Tricyclic pyrido-carboxamide derivatives as rock inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2018-03-13 US disclosed
US-7189728-B2 Inhibitors of dipeptidyl peptidase IV FERRING, BV (NL) 2007-03-13 US disclosed
US-7189728-B2 Inhibitors of dipeptidyl peptidase IV FERRING, BV (NL) 2007-03-13 US disclosed