SCHEMBL14569124

SCHEMBL14569124

O=c1[nH]c2cnc(NCCc3ccccc3F)nc2n1-c1cccc(O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.45
ADORA2A P29274 7/20 0.40
ADORA1 P30542 7/20 0.40
GPR84 Q9NQS5 1/20 0.39
RPS6KA3 P51812 1/20 0.38
MAP3K11 Q16584 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
TYRO3 Q06418 1/20 0.36
TP53 P04637 2/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
PRKCQ Q04759 1/20 0.36
FFAR1 O14842 1/20 0.36
MAPT P10636 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4507899 0.88 ADORA2A (0.53) GSK3BADORA2AADORA1USP2ALDH1A1
SCHEMBL18542913 0.77 ALDH1A1 (0.44) ADORA2AADORA1GPR84SMN1; SMN2TP53
SCHEMBL12371760 0.73 GSK3B (0.45) GSK3BADORA2AADORA1SMN1; SMN2PRKCQ
SCHEMBL12371740 0.73 GSK3B (0.45) GSK3BADORA2AADORA1SMN1; SMN2MAPT
SCHEMBL14569129 0.70 ADORA2A (0.44) GSK3BADORA2AADORA1SMN1; SMN2MAPT
SCHEMBL4512221 0.70 ADORA2A (0.63) ADORA2AADORA1TP53MEN1USP2
SCHEMBL12371703 0.69 JAK2 (0.44) ADORA2AADORA1JAK2JAK3MAPT
SCHEMBL14569011 0.69 ADORA2A (0.68) ADORA2AADORA1
SCHEMBL16034402 0.69 CASP1 (0.41) ADORA2AADORA1GPR84SMN1; SMN2MEN1
SCHEMBL18542929 0.69 MEN1 (0.44) GSK3BGPR84TP53PRKCQFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007035873-A1 PURINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES PHARMACOPEIA, INC. (US) 2007-03-29 WO disclosed