SCHEMBL14572003

SCHEMBL14572003

CCC(C)c1c(C)nc2ncccn12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 0.49
KDM4E B2RXH2 10/20 0.49
HPGD P15428 8/20 0.49
HSD17B10 Q99714 1/20 0.49
PDE1A P54750 3/20 0.37
PDE1B Q01064 3/20 0.37
PDE1C Q14123 3/20 0.37
GAA P10253 6/20 0.36
MAPT P10636 4/20 0.36
LMNA P02545 3/20 0.36
MAPK1 P28482 2/20 0.36
HTT P42858 2/20 0.36
RAB9A P51151 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALOX12 P18054 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12146430 0.83 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL19954252 0.73 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL22995769 0.72 BACE1 (0.44) ALDH1A1KDM4EHPGDHSD17B10PKM
SCHEMBL259599 0.72 KDM4E (0.51) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL23429123 0.70 ALDH1A1 (0.40) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL11892541 0.70 ALDH1A1 (0.38) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL23131729 0.70 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL13370818 0.69 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL17224054 0.69 KDM4E (0.54) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL18575691 0.69 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDHSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7196095-B2 (Pyrimidinyl) (phenyl) substituted fused heteroaryl p38 inhibiting and PKG kinase inhibiting compounds MERCK & CO., INC. (US) 2007-03-27 US disclosed