SCHEMBL14589053

SCHEMBL14589053

COC(=O)c1ccc(N)c2ccncc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.64
KDM4E B2RXH2 6/20 0.64
GAA P10253 5/20 0.64
GLA P06280 3/20 0.64
HSD17B10 Q99714 4/20 0.50
HPGD P15428 3/20 0.50
CASP1 P29466 2/20 0.50
CASP7 P55210 2/20 0.50
HTT P42858 1/20 0.50
NCOA1 Q15788 1/20 0.50
RCE1 Q9Y256 1/20 0.50
NCOA3 Q9Y6Q9 1/20 0.50
EP300 Q09472 1/20 0.47
KAT2B Q92831 1/20 0.47
KAT8 Q9H7Z6 1/20 0.47
MAPT P10636 3/20 0.45
ATM Q13315 1/20 0.45
CFTR P13569 3/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
ABL1 P00519 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21801051 0.83 KDM4E (0.53) ALDH1A1KDM4EGAAGLAHSD17B10
SCHEMBL21801064 0.81 KDM4E (0.51) ALDH1A1KDM4EGAAGLAHSD17B10
SCHEMBL28892677 0.81 KDM4E (0.51) ALDH1A1KDM4EGAAGLAHSD17B10
SCHEMBL28892356 0.81 KDM4E (0.51) ALDH1A1KDM4EGAAGLAHSD17B10
SCHEMBL30757324 0.81 KDM4E (0.51) ALDH1A1KDM4EGAAGLAHSD17B10
SCHEMBL14589054 0.80 KDM4E (0.59) ALDH1A1KDM4EGAAGLAHTT
SCHEMBL1062129 0.78 ALDH1A1 (0.74) ALDH1A1KDM4EGAAGLAHSD17B10
SCHEMBL31758437 0.78 ALDH1A1 (0.61) ALDH1A1KDM4EGAAGLAHSD17B10
SCHEMBL30419031 0.78 ALDH1A1 (0.74) ALDH1A1KDM4EGAAGLAHSD17B10
SCHEMBL29464551 0.78 ALDH1A1 (1.00) ALDH1A1KDM4EGAAGLAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7183411-B2 Naphthol, quinoline and isoquinoline-derived urea modulators of vanilloid VR1 receptor JANSSEN PHARMACEUTICA N.V. (BE) 2007-02-27 US disclosed
US-7183411-B2 Naphthol, quinoline and isoquinoline-derived urea modulators of vanilloid VR1 receptor JANSSEN PHARMACEUTICA N.V. (BE) 2007-02-27 US disclosed