SCHEMBL14589072

SCHEMBL14589072

COC(=O)c1ccc(-c2cnc(-c3cccc(I)c3)s2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 3/20 0.48
HSD17B2 P37059 3/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
SGK1 O00141 1/20 0.43
CAMKK2 Q96RR4 1/20 0.43
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
HPGD P15428 1/20 0.42
CDK8 P49336 1/20 0.41
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
PGGT1B P53609 1/20 0.41
NEK1 Q96PY6 1/20 0.41
AXL P30530 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4256137 0.81 MMP2 (0.52) HSD17B1HSD17B2CYP3A4CYP2C9MEN1
SCHEMBL7394802 0.81 CA1 (0.56) HSD17B1HSD17B2CYP3A4CYP2C9KDM4E
SCHEMBL7392985 0.80 MMP2 (0.57) KDM4ELMNAMAPTALDH1A1MEN1
SCHEMBL1505315 0.77 HSD17B1 (0.46) HSD17B1HSD17B2CYP3A4CYP2C9KDM4E
SCHEMBL28968146 0.76 CDK8 (0.51) KDM4ELMNAMAPTCDK8NEK1
SCHEMBL21873453 0.74 MAPT (0.51) KDM4ELMNAMAPTALDH1A1MEN1
SCHEMBL29016894 0.74 NEK1 (0.50) HSD17B1HSD17B2CYP3A4CYP2C9SGK1
SCHEMBL4264131 0.74 PLAU (0.52) CYP3A4MAPTALDH1A1GAAKMT2A
SCHEMBL13949639 0.73 EGFR (0.43) SGK1CAMKK2KDM4EALDH1A1EGFR
SCHEMBL15051048 0.73 CSNK2A1 (0.68) CYP3A4CYP2C9KDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179822-B2 Hetero biaryl derivatives as matrix metalloproteinase inhibitors WARNER-LAMBERT COMPANY (US) 2007-02-20 US disclosed