SCHEMBL14608901

SCHEMBL14608901

Bc1ccc2[nH]c3c(c2c1)CC(=C)N(CC(=O)OC(C)(C)C)c1ccccc1-3

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 7/20 0.52
GSK3B P49841 5/20 0.47
CCNB2 O95067 5/20 0.47
CCNB1 P14635 5/20 0.47
CCNB3 Q8WWL7 5/20 0.47
CDK5 Q00535 1/20 0.47
CDK5R1 Q15078 1/20 0.47
MDH2 P40926 14/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237362 0.79 CDK1 (0.81) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5688353 0.69 CDK1 (1.00) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL19353002 0.65 CA1 (0.69) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5235565 0.64 CDK1 (0.79) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL7091522 0.63 ALDH1A1 (0.67)
SCHEMBL12856385 0.62 CCNB2 (0.75) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL5233378 0.61 CDK1 (0.76) CDK1GSK3BCCNB2CCNB1CCNB3
SCHEMBL24714971 0.61 ALDH1A1 (0.60)
SCHEMBL5966758 0.60 CCKBR (0.48)
SCHEMBL5237969 0.59 CDK1 (0.70) CDK1GSK3BCCNB2CCNB1CCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1757607-A1 N5-substituted benzo¬2,3|azepino¬4,5-b|indol-6-ones for treating tropical diseases Molisa GmbH (DE) 2007-02-28 EP disclosed