SCHEMBL14608917

SCHEMBL14608917

Cc1cccnc1N1CCN(CC(=O)N2CCN(C3CCC3)CC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.47
ALDH1A1 P00352 5/20 0.46
KDM4E B2RXH2 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
TRPV1 Q8NER1 4/20 0.46
PARP1 P09874 2/20 0.45
MAPT P10636 3/20 0.43
TP53 P04637 1/20 0.43
KDM2B Q8NHM5 1/20 0.42
NPSR1 Q6W5P4 2/20 0.42
HTT P42858 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005240 0.87 HRH3 (0.49) HRH3ALDH1A1KDM4ETDP1PARP1
SCHEMBL13005239 0.85 HRH3 (0.47) HRH3ALDH1A1KDM4ETDP1PARP1
SCHEMBL3771811 0.85 HRH3 (0.67) HRH3ALDH1A1TRPV1MAPTNPSR1
SCHEMBL3772561 0.83 ALDH1A1 (0.52) HRH3ALDH1A1KDM4EPARP1MAPT
SCHEMBL3776097 0.82 HRH3 (0.64) HRH3ALDH1A1KDM4ETRPV1MAPT
SCHEMBL3767997 0.82 TSHR (0.53) ALDH1A1KDM4ETDP1MAPTTP53
SCHEMBL3774250 0.81 MAPT (0.60) ALDH1A1KDM4EMAPTNPSR1HTT
SCHEMBL3771221 0.81 ALDH1A1 (0.52) ALDH1A1KDM4EPARP1MAPTNPSR1
SCHEMBL13004952 0.81 KDM4E (0.67) ALDH1A1KDM4ETDP1PARP1MAPT
SCHEMBL3765753 0.80 ALDH1A1 (0.52) ALDH1A1KDM4EPARP1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007016496-A2 DIPIPERAZINYL KETONES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2007-02-08 WO disclosed