SCHEMBL14609883

SCHEMBL14609883

COCC(c1nc(O)c(O)c(C(=O)NCc2ccc(F)cc2)n1)N(C)CI

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNE1 P15382 1/20 0.41
CCR1 P32246 1/20 0.41
KCNQ1 P51787 1/20 0.41
POLB P06746 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ERCC1 P07992 1/20 0.38
FEN1 P39748 1/20 0.38
ERCC4 Q92889 1/20 0.38
KCNH2 Q12809 1/20 0.38
CYP2C9 P11712 1/20 0.38
ALDH1A1 P00352 4/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
KCNQ3 O43525 1/20 0.37
KCNQ2 O43526 1/20 0.37
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5121784 0.90 KCNE1 (0.43) KCNE1CCR1KCNQ1POLBSMN1; SMN2
SCHEMBL5127902 0.88 KCNE1 (0.41) KCNE1CCR1KCNQ1POLBSMN1; SMN2
SCHEMBL5248354 0.83 KCNE1 (0.43) KCNE1CCR1KCNQ1POLBSMN1; SMN2
SCHEMBL5124916 0.82 KCNE1 (0.44) KCNE1CCR1KCNQ1POLBSMN1; SMN2
SCHEMBL5124165 0.81 POLB (0.42) KCNE1CCR1KCNQ1POLBSMN1; SMN2
SCHEMBL5128685 0.81 ALDH1A1 (0.39) KCNE1CCR1KCNQ1POLBSMN1; SMN2
SCHEMBL5122432 0.80 KCNE1 (0.42) KCNE1CCR1KCNQ1POLBSMN1; SMN2
SCHEMBL5252830 0.80 EGLN1 (0.44) KCNE1CCR1KCNQ1POLBSMN1; SMN2
SCHEMBL5123957 0.80 ALDH1A1 (0.43) POLBSMN1; SMN2ERCC1FEN1ERCC4
SCHEMBL5114416 0.79 SMN1; SMN2 (0.40) KCNE1CCR1KCNQ1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441734-B1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ANGELETTI P IST RICHERCHE BIO (IT) 2007-02-28 EP disclosed