SCHEMBL14616447

SCHEMBL14616447

O=CCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCC=O

nearest known ligand 0.75

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.75
TSHR P16473 2/20 0.69
FAAH O00519 2/20 0.58
TRPV1 Q8NER1 2/20 0.58
ALDH1A1 P00352 2/20 0.44
TDP1 Q9NUW8 2/20 0.37
MAPK1 P28482 1/20 0.33
MAPT P10636 1/20 0.32
EPHX1 P07099 1/20 0.32
ADH1B P00325 1/20 0.32
ADH1C P00326 1/20 0.32
ADH1A P07327 1/20 0.32
ADH4 P08319 1/20 0.32
ADH7 P40394 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2153681 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1
SCHEMBL14337652 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1
SCHEMBL495540 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1
SCHEMBL3227000 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1
SCHEMBL1676895 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1
SCHEMBL17369100 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1
SCHEMBL1489327 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1
SCHEMBL1676795 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1
SCHEMBL2153965 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1
SCHEMBL2155121 1.00 HIF1A (0.75) HIF1ATSHRFAAHTRPV1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10000447-B2 Compounds for targeting drug delivery and enhancing siRNA activity NITTO DENKO CORPORATION (JP) 2018-06-19 US disclosed
US-20170000893-A1 COMPOUNDS FOR TARGETING DRUG DELIVERY AND ENHANCING siRNA ACTIVITY NITTO DENKO CORP (JP) 2017-01-05 US disclosed
US-20170001950-A1 COMPOUNDS FOR TARGETING DRUG DELIVERY AND ENHANCING siRNA ACTIVITY NITTO DENKO CORP (JP) 2017-01-05 US disclosed
US-20160263254-A1 TARGETING VECTOR-PHOSPHOLIPID CONJUGATES BRACCO INTERNATIONAL B.V. (NL) 2016-09-15 US disclosed
US-9393315-B2 Compounds for targeting drug delivery and enhancing siRNA activity NITTO DENKO CORPORATION (JP) 2016-07-19 US disclosed
US-20140294973-A1 PHARMACEUTICAL COMPOSITIONS OF HYDROPHOBIC CAMPTOTHECIN DERIVATIVES TAIWAN LIPOSOME COMPANY, LTD. (TW) 2014-10-02 US disclosed
US-20130017249-A1 COMPOUNDS FOR TARGETING DRUG DELIVERY AND ENHANCING siRNA ACTIVITY NITTO DENKO CORPORATION (JP) 2013-01-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140294973-A1 PHARMACEUTICAL COMPOSITIONS OF HYDROPHOBIC CAMPTOTHECIN DERIVATIVES PTEN, LIPA, PHOSPHO1 HIF1A 1780/4885TSHR 3384/4885FAAH 2338/4885
US-20160263254-A1 TARGETING VECTOR-PHOSPHOLIPID CONJUGATES KDR, FLT4, PTAFR HIF1A 698/4885TSHR 1302/4885FAAH 924/4885
US-20130017249-A1 COMPOUNDS FOR TARGETING DRUG DELIVERY AND ENHANCING siRNA ACTIVITY LDLR, RARG, FABP4 HIF1A 3069/4885TSHR 1224/4885FAAH 1316/4885
US-10000447-B2 Compounds for targeting drug delivery and enhancing siRNA activity LDLR, RARG, FABP4 HIF1A 3069/4885TSHR 1224/4885FAAH 1316/4885
US-20170001950-A1 COMPOUNDS FOR TARGETING DRUG DELIVERY AND ENHANCING siRNA ACTIVITY LDLR, RARG, FABP4 HIF1A 3069/4885TSHR 1224/4885FAAH 1316/4885
US-20170000893-A1 COMPOUNDS FOR TARGETING DRUG DELIVERY AND ENHANCING siRNA ACTIVITY LDLR, RARG, FABP4 HIF1A 3069/4885TSHR 1224/4885FAAH 1316/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.