SCHEMBL1461804

SCHEMBL1461804

CC(C)(C)N(Cc1cn(CCON2C(=O)c3ccccc3C2=O)nn1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 4/20 0.47
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 1/20 0.38
CYP1A2 P05177 2/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP2C9 P11712 1/20 0.37
RECQL P46063 1/20 0.37
ABCG2 Q9UNQ0 4/20 0.36
MAOB P27338 1/20 0.35
ABCC1 P33527 3/20 0.35
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
ABCB1 P08183 1/20 0.35
TYR P14679 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1461599 0.82 HSP90AB1 (0.39) HSP90AB1MEN1NPC1RAB9AKMT2A
SCHEMBL12275366 0.78 GAA (0.42) HSP90AB1L3MBTL1GAACYP1A2ALDH1A1
SCHEMBL12275365 0.78 HSP90AB1 (0.45) HSP90AB1L3MBTL1GAACYP1A2ALDH1A1
SCHEMBL12451342 0.77 CA1 (0.46) HSP90AB1GAAALDH1A1RECQL
SCHEMBL18839649 0.77 HSP90AB1 (0.49) HSP90AB1MEN1KMT2AGAAALDH1A1
SCHEMBL16714956 0.76 MEN1 (0.50) MEN1NPC1RAB9AKMT2AL3MBTL1
SCHEMBL1461801 0.73 GAA (0.38) HSP90AB1MEN1KMT2AGAACYP1A2
SCHEMBL20518699 0.72 GAA (0.40) HSP90AB1MEN1RAB9AKMT2AGAA
SCHEMBL25214310 0.71 HSP90AB1 (0.37) HSP90AB1MEN1NPC1RAB9AKMT2A
SCHEMBL1461856 0.71 GAA (0.40) HSP90AB1MEN1KMT2AGAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011029639-A2 COMPOUNDS AND METHODS FOR TREATING NEOPLASIA MEDEXIS S.A. (GR) 2011-03-17 WO disclosed