SCHEMBL1461801

SCHEMBL1461801

CC(C)(C)C(NC(=O)O)c1cn(CCON2C(=O)c3ccccc3C2=O)nn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 1/20 0.37
RECQL P46063 1/20 0.37
HSP90AB1 P08238 2/20 0.36
MDM2 Q00987 1/20 0.35
XIAP P98170 2/20 0.34
BIRC3 Q13489 2/20 0.34
BIRC2 Q13490 2/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HDAC3 O15379 2/20 0.33
HDAC4 P56524 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC7 Q8WUI4 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC10 Q969S8 2/20 0.33
HDAC11 Q96DB2 2/20 0.33
HDAC8 Q9BY41 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1461597 0.83 PDE4A (0.35) ALDH1A1CYP1A2CYP2C9HSP90AB1KMT2A
SCHEMBL1461856 0.81 GAA (0.40) GAAALDH1A1CYP1A2CYP2C9RECQL
SCHEMBL12275365 0.75 HSP90AB1 (0.45) GAAALDH1A1CYP1A2CYP2C9RECQL
SCHEMBL1461804 0.73 HSP90AB1 (0.47) GAAALDH1A1CYP1A2CYP2C9RECQL
SCHEMBL12275366 0.73 GAA (0.42) GAAALDH1A1CYP1A2CYP2C9RECQL
SCHEMBL4267815 0.73 GAA (0.47) GAAALDH1A1CYP1A2CYP2C9RECQL
SCHEMBL12451342 0.73 CA1 (0.46) GAAALDH1A1RECQLHSP90AB1POLB
SCHEMBL18839649 0.72 HSP90AB1 (0.49) GAAALDH1A1RECQLHSP90AB1KMT2A
SCHEMBL20518699 0.69 GAA (0.40) GAAALDH1A1CYP1A2CYP2C9RECQL
SCHEMBL26347332 0.67 DGAT1 (0.51) ALDH1A1HSP90AB1MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011029639-A2 COMPOUNDS AND METHODS FOR TREATING NEOPLASIA MEDEXIS S.A. (GR) 2011-03-17 WO disclosed