SCHEMBL14619

SCHEMBL14619

Cc1cc(-c2cc(=O)n3cc(-c4ccc(CNCCCN)cc4)c(=O)nc3[nH]2)ccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.38
ENPP2 Q13822 1/20 0.33
CNR1 P21554 2/20 0.31
MC4R P32245 1/20 0.31
MC5R P33032 1/20 0.31
MC3R P41968 1/20 0.31
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
VSIR Q9H7M9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11960641 0.92 MARS1 (0.33) CNR2MC4RMC5RMC3R
SCHEMBL20124187 0.91 MC4R (0.32) MC4RMC5RMC3R
SCHEMBL11960637 0.86 PDCD1 (0.37) MC4RMC5RMC3RKDM4ENPC1
SCHEMBL19573483 0.85 MC4R (0.34) MC4RMC5RMC3R
SCHEMBL14613 0.85 MC4R (0.34) MC4RMC5RMC3R
SCHEMBL11960639 0.84 CHRM2 (0.38) MC4RMC5RMC3RKDM4EALDH1A1
SCHEMBL20124107 0.84 HDAC1 (0.34) CNR1MC4RMC5RMC3RVSIR
SCHEMBL11960642 0.83 HDAC1 (0.34) MC4RMC5RMC3R
SCHEMBL11208 0.82 MC4R (0.33) MC4RMC5RMC3R
SCHEMBL11960640 0.82 MAP3K11 (0.35) KDM4EPDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488532-B1 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME MELINTA THERAPEUTICS INC (US) 2018-05-09 EP disclosed
WO-2011047320-A2 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME RIB-X PHARMACEUTICALS, INC. (US) 2011-04-21 WO disclosed