SCHEMBL14619906

SCHEMBL14619906

CC(=O)OCCOc1ccc(S(=O)(=O)N2CCSC(C)(C)[C@@H]2C(=O)NO)cc1

nearest known ligand 0.81

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 20/20 0.81
MMP13 P45452 19/20 0.81
ADAM17 P78536 15/20 0.81
MMP3 P08254 8/20 0.74
MMP2 P08253 7/20 0.74
MMP7 P09237 5/20 0.74
MMP9 P14780 7/20 0.72
MMP8 P22894 3/20 0.72
ADAM10 O14672 2/20 0.70
ADAM9 Q13443 2/20 0.70
MMP14 P50281 2/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3947996 0.88 MMP1 (0.83) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL8394315 0.88 MMP1 (0.62) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL3945461 0.86 MMP1 (0.82) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL6383433 0.86 MMP1 (0.77) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL7075595 0.85 MMP1 (0.75) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL7351911 0.84 MMP1 (1.00) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL3948482 0.84 MMP1 (1.00) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL8033898 0.84 MMP1 (0.80) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL2358255 0.83 ADAM17 (1.00) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL3942486 0.83 ADAM17 (1.00) MMP1MMP13ADAM17MMP3MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179911-B2 coupling a silyl ester of (3S)-2,2-dimethyl-tetrahydro-2H-1,4-thiazine-3-carboxylic acid with 6,4-[4-(chlorosulfonyl)phenoxy]-2-butynyl acetate, hydrolyzing the silyl ester WYETH (US) 2007-02-20 US disclosed