SCHEMBL1462495

SCHEMBL1462495

CCCCCOc1ccnc2c(C(F)(F)F)cccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.43
NR1H2 P55055 3/20 0.43
NR1H3 Q13133 3/20 0.43
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
MCHR1 Q99705 2/20 0.41
PARP1 P09874 1/20 0.40
CNR1 P21554 2/20 0.40
CNR2 P34972 2/20 0.40
CYP2C9 P11712 1/20 0.40
MEN1 O00255 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC2A1 P11166 1/20 0.39
S1PR1 P21453 1/20 0.39
KCNH2 Q12809 2/20 0.38
RXRA P19793 1/20 0.38
HTR1B P28222 1/20 0.38
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8271684 0.79 NCF1 (0.49) NCF1NR1H2NR1H3PARP1RXRA
SCHEMBL348618 0.79 HTR1A (0.57) MCHR1CNR1CNR2MEN1HTT
SCHEMBL13045005 0.79 NCF1 (0.44) NCF1NR1H2NR1H3PARP1HTT
SCHEMBL17018214 0.79 MCHR1 (0.44) MCHR1CNR1CNR2CYP2C9MEN1
SCHEMBL15923479 0.78 HTR1A (0.53) HTTKCNH2DYRK3PRKD3MAP4K4
SCHEMBL11011220 0.78 NCF1 (0.48) NCF1NR1H2NR1H3ADORA2AADORA1
SCHEMBL10203093 0.77 NR1H2 (0.43) NCF1NR1H2NR1H3ADORA2AADORA1
SCHEMBL1091092 0.77 KDM4E (0.49) NCF1NR1H2NR1H3PARP1DYRK3
SCHEMBL16234628 0.77 GSK3A (0.45) NCF1NR1H2NR1H3ADORA2AADORA1
SCHEMBL13409380 0.75 NCF1 (0.46) NCF1NR1H2NR1H3PARP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4648894-B2 2011-03-09 JP claimed
JP-2006519221-A 2006-08-24 JP claimed
EP-1597253-A2 COMPOUNDS AND METHODS OF TREATING CELL PROLIFERATIVE DISEASES, RETINOPATHIES AND ARTHRITIS Exonhit Therapeutics S.A. (FR) 2005-11-23 EP claimed
WO-2004076445-A2 COMPOUNDS AND METHODS OF TREATING CELL PROLIFERATIVE DISEASES, RETINOPATHIES AND ARTHRITIS EXONHIT THERAPEUTICS SA (FR) 2004-09-10 WO claimed