SCHEMBL14629978

SCHEMBL14629978

c1cc2nc(C3CC3)ccc2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 5/20 0.37
PAK4 O96013 1/20 0.37
IDO1 P14902 1/20 0.36
PAK3 O75914 3/20 0.35
PAK2 Q13177 3/20 0.35
TRPA1 O75762 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ITGB2 P05107 1/20 0.34
ICAM1 P05362 1/20 0.34
ITGAL P20701 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
AHR P35869 1/20 0.34
ADK P55263 1/20 0.34
MAOB P27338 4/20 0.33
POLB P06746 1/20 0.33
PRMT5 O14744 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30587475 0.72 ROCK2 (0.44) PAK4IDO1TRPA1POLBKDM4E
SCHEMBL12855676 0.71
SCHEMBL14630025 0.71 AXL (0.39) TRPA1CA1CA2ITGB2ICAM1
SCHEMBL31252444 0.70 CHRNA7 (0.35) PAK1PAK4TRPA1CA1CA2
SCHEMBL7622138 0.69 ALDH1A1 (0.33) POLBKDM4EMAPTTSHRHSD17B10
SCHEMBL19212577 0.69 IDO1 (0.42) IDO1MAOBPOLBPRMT5KCNH2
SCHEMBL2352863 0.68 SYK (0.33) POLBMAPTHSD17B10MAPK8MAPK10
SCHEMBL9377967 0.68 JAK3 (0.40) JAK2
SCHEMBL23625710 0.67 APP (0.44) TRPA1CA1CA2ITGB2ICAM1
SCHEMBL7016588 0.67 USP2 (0.43) TRPA1CA1CA2ITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2548876-A1 New CRTh2 antagonists Almirall, S.A. (ES) 2013-01-23 EP disclosed