SCHEMBL14635929

SCHEMBL14635929

CCCc1cccnc1NC(=O)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.60
NPC1 O15118 5/20 0.56
RAB9A P51151 5/20 0.56
L3MBTL1 Q9Y468 1/20 0.54
ATM Q13315 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
KDR P35968 1/20 0.47
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
ADORA3 P0DMS8 2/20 0.46
TRPV1 Q8NER1 1/20 0.46
PABPC1 P11940 1/20 0.45
GRM5 P41594 1/20 0.45
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23566407 0.91 HTT (0.63) HTTNPC1RAB9AATMMEN1
SCHEMBL28018732 0.84 GRM5 (0.52) HTTNPC1RAB9AL3MBTL1ATM
SCHEMBL6176906 0.83 HTT (0.54) HTTNPC1RAB9AATMMEN1
SCHEMBL16244495 0.80 KDM4E (0.50) NPC1RAB9AL3MBTL1MAPTGRM5
SCHEMBL6174461 0.79 HTT (0.56) HTTNPC1RAB9AL3MBTL1ATM
SCHEMBL19426861 0.78 KDM4E (0.55) HTTNPC1RAB9AL3MBTL1MEN1
SCHEMBL7532358 0.78 KMT2A (0.68) HTTNPC1RAB9AL3MBTL1ATM
SCHEMBL12844413 0.78 GRM5 (0.46) NPC1RAB9AL3MBTL1GRM5
SCHEMBL30648563 0.76 RAB9A (0.88) HTTNPC1RAB9AATMMEN1
SCHEMBL3364009 0.76 MME (0.52) HTTNPC1RAB9AL3MBTL1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2734529-A1 BTK INHIBITORS Merck Sharp & Dohme Corp. (US) 2014-05-28 EP disclosed
WO-2013010380-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-01-24 WO disclosed