SCHEMBL14636120

SCHEMBL14636120

CC(C)(C)OC(=O)N1CC=C(c2cccc(-c3nnn[nH]3)c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.51
GRM1 Q13255 11/20 0.49
GRM5 P41594 10/20 0.49
PDK4 Q16654 1/20 0.49
CDK7 P50613 1/20 0.46
CDK13 Q14004 1/20 0.46
CDK12 Q9NYV4 1/20 0.46
SOS1 Q07889 1/20 0.45
CYP11B2 P19099 1/20 0.45
JAK1 P23458 1/20 0.43
CDK9 P50750 1/20 0.42
CNR1 P21554 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2811392 0.82 PDK4 (0.60) NAMPTGRM1GRM5PDK4CYP11B2
SCHEMBL7831576 0.81 PDK4 (0.58) NAMPTGRM1GRM5PDK4CDK7
SCHEMBL29914645 0.80 PDK4 (0.57) NAMPTGRM1GRM5PDK4SOS1
SCHEMBL1364792 0.80 PDK4 (0.57) NAMPTGRM1GRM5PDK4SOS1
SCHEMBL13994079 0.79 CDK9 (0.47) NAMPTGRM1GRM5CDK9
SCHEMBL14500280 0.79 CDK9 (0.54) CDK9
SCHEMBL2239831 0.79 NAMPT (0.66) NAMPTGRM1GRM5PDK4
SCHEMBL4459006 0.79 PDK4 (0.54) NAMPTGRM1GRM5PDK4CDK7
SCHEMBL3988457 0.79 PDK4 (0.56) NAMPTGRM1GRM5PDK4CDK7
SCHEMBL13261659 0.79 PDK4 (0.56) NAMPTGRM1GRM5PDK4CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013010453-A1 CHEMOKING RECEPTOR ANTAGONISTS ABBOTT LABORATORIES (US) 2013-01-24 WO disclosed