SCHEMBL14636633

SCHEMBL14636633

O=C(Nc1ccccn1)c1ccccc1F

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.69
KMT2A Q03164 4/20 0.69
KDM4E B2RXH2 2/20 0.69
L3MBTL1 Q9Y468 1/20 0.69
NPC1 O15118 6/20 0.64
RAB9A P51151 6/20 0.64
SMN1; SMN2 Q16637 4/20 0.64
GAA P10253 4/20 0.64
TP53 P04637 2/20 0.64
TDP1 Q9NUW8 2/20 0.64
ALDH1A1 P00352 1/20 0.64
GLA P06280 1/20 0.64
HSD17B10 Q99714 1/20 0.64
CHRNB2 P17787 1/20 0.63
CHRNB4 P30926 1/20 0.63
CHRNA3 P32297 1/20 0.63
CHRNA4 P43681 1/20 0.63
HTT P42858 1/20 0.59
PKM P14618 1/20 0.58
SGMS2 Q8NHU3 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30362638 1.00 MEN1 (0.69) MEN1KMT2AKDM4EL3MBTL1NPC1
SCHEMBL30643216 0.89 MEN1 (0.63) MEN1KMT2AKDM4EL3MBTL1NPC1
SCHEMBL6815217 0.85 KMT2A (0.61) MEN1KMT2AKDM4EL3MBTL1NPC1
SCHEMBL27487339 0.84 MEN1 (0.57) MEN1KMT2AKDM4EL3MBTL1NPC1
SCHEMBL8129469 0.84 MEN1 (0.57) MEN1KMT2AKDM4EL3MBTL1NPC1
SCHEMBL20332736 0.82 SORT1 (0.71) MEN1KMT2AKDM4EL3MBTL1NPC1
SCHEMBL17675194 0.81 MEN1 (0.71) MEN1KMT2AKDM4EL3MBTL1NPC1
SCHEMBL8433498 0.81 MEN1 (1.00) MEN1KMT2AKDM4EL3MBTL1NPC1
SCHEMBL23446474 0.80 SMN1; SMN2 (0.56) MEN1KMT2AKDM4ENPC1RAB9A
SCHEMBL1966818 0.80 SMN1; SMN2 (0.64) MEN1KMT2AKDM4EL3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113735850-A Synthesis method of 1,2, 4-triazole compound 河南师范大学 2021-12-03 CN disclosed
EP-2734529-A1 BTK INHIBITORS Merck Sharp & Dohme Corp. (US) 2014-05-28 EP disclosed
WO-2013010380-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-01-24 WO disclosed
CN-1177356-A Bicyclic benzazepine derivatives as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-03-25 CN disclosed