SCHEMBL146370

SCHEMBL146370

O=C(O)C1Cc2[nH]cnc2CN1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.46
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ADRA1A P35348 3/20 0.39
MAPT P10636 1/20 0.38
GRIA2 P42262 1/20 0.38
HTR3A P46098 2/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
SLC6A4 P31645 1/20 0.33
OPRK1 P41145 1/20 0.33
HTR2B P41595 1/20 0.33
KCNH2 Q12809 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3739922 1.00 EGLN1 (0.46) EGLN1KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL9582230 1.00 EGLN1 (0.46) EGLN1KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL3738082 0.98 EGLN1 (0.44) EGLN1KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL9582700 0.98 EGLN1 (0.44) EGLN1KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL9582091 0.98 EGLN1 (0.44) EGLN1KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL6874923 0.98 EGLN1 (0.44) EGLN1KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL3804263 0.98 EGLN1 (0.44) EGLN1KDM4EALDH1A1GAASMN1; SMN2
Trifluoroacetic Acid SCHEMBL23704593 0.91 KDM4E (0.42) EGLN1KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL10544160 0.87 EGLN1 (0.46) EGLN1KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL10544179 0.87 EGLN1 (0.46) EGLN1KDM4EALDH1A1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 388 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12428447-B2 Peptide-based non-proteinaceous cargo delivery FELDAN BIO INC. (CA) 2025-09-30 US claimed
US-20240197896-A1 SYNTHETIC PEPTIDE SHUTTLE AGENT BIOCONJUGATES FOR INTRACELLULAR CARGO DELIVERY FELDAN BIO INC. (CA) 2024-06-20 US claimed
EP-4313159-A1 SYNTHETIC PEPTIDE SHUTTLE AGENT BIOCONJUGATES FOR INTRACELLULAR CARGO DELIVERY Feldan Bio Inc. (CA) 2024-02-07 EP claimed
US-20230399661-A1 SHUTTLE AGENT PEPTIDES OF MINIMAL LENGTH AND VARIANTS THEREOF ADAPTED FOR TRANSDUCTION OF CAS9-RNP AND OTHER NUCLEOPROTEIN CARGOS FELDAN BIO INC. (CA) 2023-12-14 US claimed
US-20230383291-A1 PEPTIDE-BASED TRANSDUCTION OF NON-ANIONIC POLYNUCLEOTIDE ANALOGS FOR GENE EXPRESSION MODULATION FELDAN BIO INC. (CA) 2023-11-30 US claimed
EP-4232590-A1 SHUTTLE AGENT PEPTIDES OF MINIMAL LENGTH AND VARIANTS THEREOF ADAPTED FOR TRANSDUCTION OF CAS9-RNP AND OTHER NUCLEOPROTEIN CARGOS Feldan Bio Inc. (CA) 2023-08-30 EP claimed
EP-4229207-A1 PEPTIDE-BASED TRANSDUCTION OF NON-ANIONIC POLYNUCLEOTIDE ANALOGS FOR GENE EXPRESSION MODULATION Feldan Bio Inc. (CA) 2023-08-23 EP claimed
WO-2022204806-A1 SYNTHETIC PEPTIDE SHUTTLE AGENT BIOCONJUGATES FOR INTRACELLULAR CARGO DELIVERY FELDAN BIO INC. (CA) 2022-10-06 WO claimed
US-20220204561-A1 PEPTIDE-BASED NON-PROTEINACEOUS CARGO DELIVERY FELDAN BIO INC. (CA) 2022-06-30 US claimed
WO-2022082315-A1 SHUTTLE AGENT PEPTIDES OF MINIMAL LENGH AND VARIANTS THEREOF ADAPTED FOR TRANSDUCTION OF CAS9-RNP AND OTHER NUCLEOPROTEIN CARGOS FELDAN BIO INC. (CA) 2022-04-28 WO claimed
US-20190070153-A1 COMPOSITIONS AND METHODS FOR TREATING PULMONARY DISEASES CASE WESTERN RESERVE UNIVERSITY 2019-03-07 US claimed
US-20180200233-A1 COMPOSITIONS FOR PREVENTING CANCERS ASSOCIATED WITH HUMAN PAPILLOMA VIRUSES LOMA LINDA UNIVERSITY 2018-07-19 US claimed
EP-3322418-A1 COMPOSITIONS FOR PREVENTING CANCERS ASSOCIATED WITH HUMAN PAPILLOMA VIRUSES Loma Linda University (US) 2018-05-23 EP claimed
WO-2017062988-A1 COMPOSITIONS AND METHODS FOR TREATING PULMONARY DISEASES CASE WESTERN RESERVE UNIVERSITY (US) 2017-04-13 WO claimed
WO-2017011473-A1 COMPOSITIONS FOR PREVENTING CANCERS ASSOCIATED WITH HUMAN PAPILLOMA VIRUSES LOMA LINDA UNIVERSITY (US) 2017-01-19 WO claimed
US-6251280-B1 A TEMPLATE MOLECULE IS BOUND TO ONE END OF BIFUNCTIONAL LIGANDS TO FORM A COMPLEX PRIOR TO BINDING OF THE BIFUNCTIONAL LIGANDS TO THE SUBSTRATE. UNIVERSITY OF TENNESSEE RESEARCH CORPORATION 2001-06-26 US claimed
US-5317014-A Analgesics, antiinflammatory agents, antagonist, antiallergens or gastrointestinal disorders ADIR ET COMPAGNIE (FR) 1994-05-31 US claimed
US-5262537-A Treatment of nausea and vomiting ANAQUEST, INC. (US) 1993-11-16 US claimed
EP-0517589-A2 Tachykinin derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-12-09 EP claimed
EP-0104041-B1 ENZYME INHIBITORS Aktiebolaget Hässle (SE) 1988-07-27 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190070153-A1 COMPOSITIONS AND METHODS FOR TREATING PULMONARY DISEASES ACE, AGT, AGTR2 EGLN1 681/4885KDM4E 4745/4885ALDH1A1 2624/4885
US-20240197896-A1 SYNTHETIC PEPTIDE SHUTTLE AGENT BIOCONJUGATES FOR INTRACELLULAR CARGO DELIVERY SCAMP2, SLC7A1, NUMA1 EGLN1 4480/4885KDM4E 4852/4885ALDH1A1 4747/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.