SCHEMBL14642017

SCHEMBL14642017

COc1ccc(CI)c(C)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.44
KDM1A O60341 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
HTT P42858 1/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15998535 0.83 IDO1 (0.43) APLNRKMT2AALDH1A1MEN1CA12
SCHEMBL11295684 0.83 GPR84 (0.47) APLNRKDM1AMAOAMAOBKMT2A
SCHEMBL1690285 0.81 HTT (0.46) APLNRKDM1AMAOAMAOBKMT2A
SCHEMBL5177898 0.80 KMT2A (0.50) APLNRKDM1AMAOAMAOBKMT2A
SCHEMBL24411006 0.79 CA12 (0.45) APLNRKDM1AMAOAMAOBKMT2A
SCHEMBL7704446 0.79 KMT2A (0.46) APLNRKDM1AMAOAMAOBKMT2A
SCHEMBL3258877 0.79 IDO1 (0.48) APLNRKDM1AMAOAMAOBKMT2A
SCHEMBL16139667 0.79 APLNR (0.63) APLNRALDH1A1CA12CA1CA2
SCHEMBL7826059 0.79 CA12 (0.46) APLNRKDM1AMAOAMAOBKMT2A
SCHEMBL10696244 0.79 APLNR (0.44) APLNRKDM1AMAOAMAOBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8354432-B2 Cyclic derivatives as modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB COMPANY (US) 2013-01-15 US disclosed