SCHEMBL14664253

SCHEMBL14664253

O=C(O)CC(NC(=O)[C@H](Cc1ccccc1)n1cccc(NC(=O)c2c(Cl)cccc2Cl)c1=O)C(=O)CF

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.53
CASP1 P29466 19/20 0.50
CASP7 P55210 1/20 0.49
CASP8 Q14790 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL486958 1.00 CASP3 (0.53) CASP3CASP1CASP7CASP8
SCHEMBL486960 1.00 CASP3 (0.53) CASP3CASP1CASP7CASP8
SCHEMBL486962 1.00 CASP3 (0.53) CASP3CASP1CASP7CASP8
SCHEMBL5986673 0.90 CASP3 (0.53) CASP3CASP1CASP7CASP8
SCHEMBL14664252 0.90 CASP3 (0.53) CASP3CASP1CASP7CASP8
SCHEMBL5986677 0.90 CASP3 (0.53) CASP3CASP1CASP7CASP8
SCHEMBL5986681 0.90 CASP3 (0.53) CASP3CASP1CASP7CASP8
SCHEMBL473235 0.90 CASP1 (0.57) CASP3CASP1CASP7CASP8
SCHEMBL473234 0.90 CASP1 (0.57) CASP3CASP1CASP7CASP8
SCHEMBL473232 0.90 CASP1 (0.57) CASP3CASP1CASP7CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8362043-B2 Use in controlling apoptosis, as antiinflammatory agents, in treating autoimmune disease, as antiischemic agents, in treating cardiovascular disorders; for example, 3(R,S)-[2(S)-(3-Benzoylamino-2-oxo-2H-pyridin-1-yl)-3-phenyl-propionylamino]-5-fluoro-4-oxo-pentanoic acid VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-01-29 US disclosed
US-8362043-B2 Use in controlling apoptosis, as antiinflammatory agents, in treating autoimmune disease, as antiischemic agents, in treating cardiovascular disorders; for example, 3(R,S)-[2(S)-(3-Benzoylamino-2-oxo-2H-pyridin-1-yl)-3-phenyl-propionylamino]-5-fluoro-4-oxo-pentanoic acid VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-01-29 US disclosed