SCHEMBL14670282

SCHEMBL14670282

COC(=O)Nc1ccc(NC(=O)[C@H](C)N)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.62
SMN1; SMN2 Q16637 3/20 0.58
LTA4H P09960 1/20 0.54
XIAP P98170 1/20 0.52
MAPT P10636 3/20 0.50
HPGD P15428 2/20 0.50
NPC1 O15118 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
RAB9A P51151 1/20 0.49
HTT P42858 1/20 0.46
IDO1 P14902 2/20 0.45
AAK1 Q2M2I8 1/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
CIT O14578 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14670283 1.00 TAAR1 (0.62) TAAR1SMN1; SMN2LTA4HXIAPMAPT
SCHEMBL11648108 0.92 SMN1; SMN2 (0.64) TAAR1SMN1; SMN2LTA4HXIAPHPGD
SCHEMBL11644342 0.91 MEN1 (0.54) TAAR1SMN1; SMN2LTA4HXIAPMAPT
SCHEMBL11642552 0.89 CA1 (0.51) TAAR1SMN1; SMN2LTA4HXIAPMAPT
SCHEMBL11642578 0.88 TAAR1 (0.50) TAAR1SMN1; SMN2LTA4HXIAPMAPT
SCHEMBL16981649 0.84 HTT (0.66) TAAR1SMN1; SMN2LTA4HXIAPHPGD
SCHEMBL15244875 0.82 TAAR1 (0.86) TAAR1SMN1; SMN2LTA4HXIAPMAPT
SCHEMBL26347292 0.82 L3MBTL1 (0.59) TAAR1SMN1; SMN2LTA4HMAPTHPGD
SCHEMBL30503502 0.82 L3MBTL1 (0.59) TAAR1SMN1; SMN2LTA4HMAPTHPGD
SCHEMBL11641056 0.82 MTNR1B (0.60) TAAR1SMN1; SMN2LTA4HXIAPHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152664-B1 DIPEPTIDE ANALOGS AS COAGULATION FACTOR INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2014-09-03 EP disclosed
US-8367709-B2 Dipeptide analogs as coagulation factor inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2013-02-05 US disclosed