SCHEMBL14698995

SCHEMBL14698995

Cc1ccc(C(=O)N(C)c2ccc3c(c2)nc(N)n3CC(C)(C)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITK Q08881 19/20 0.49
INSR P06213 6/20 0.47
TXK P42681 2/20 0.43
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
JAK3 P52333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14708819 0.91 ITK (0.55) ITKINSRTXK
SCHEMBL14698953 0.83 ITK (0.65) ITKINSRTXK
SCHEMBL14708857 0.82 ITK (0.46) ITKINSR
SCHEMBL6274413 0.82 ITK (0.39) ITKINSRJAK2JAK1TYK2
SCHEMBL14708876 0.82 ITK (0.39) ITKINSR
SCHEMBL21310889 0.81 BACE1 (0.39) ITKINSR
SCHEMBL6415126 0.80 ITK (0.38) ITKINSR
SCHEMBL6277070 0.80 ALDH1A1 (0.38) ITKINSR
SCHEMBL21310819 0.79 TLR8 (0.58) JAK2JAK1TYK2JAK3
SCHEMBL14697486 0.78 ITK (0.49) ITKINSRTXK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013024427-A1 NOVEL UREA DERIVATIVES AS TEC KINASE INHIBITORS AND USES THEREOF GLENMARK PHARMACEUTICALS S.A. (CH) 2013-02-21 WO disclosed