SCHEMBL14699554

SCHEMBL14699554

Fc1cccc(-c2cc(-c3cccnc3)n(C3CCCCO3)n2)n1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATR Q13535 2/20 0.42
CYP4F2 P78329 4/20 0.41
CYP4A11 Q02928 4/20 0.41
PIM1 P11309 1/20 0.39
MCL1 Q07820 1/20 0.36
PDE8B O95263 1/20 0.36
CHRNB2 P17787 2/20 0.36
CHRNA6 Q15825 1/20 0.36
PIK3CD O00329 3/20 0.35
JAK1 P23458 1/20 0.35
CHRNA4 P43681 1/20 0.34
RET P07949 1/20 0.33
TNF P01375 1/20 0.33
PPARA Q07869 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP2A6 P11509 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14688866 0.79 PIM1 (0.51) ATRCYP4F2CYP4A11PIM1
SCHEMBL3433339 0.73 CYP4F2 (0.39) CYP4F2CYP4A11PIM1MCL1PDE8B
SCHEMBL14699428 0.71 IRAK4 (0.39) CYP4F2CYP4A11PIK3CDJAK1RET
SCHEMBL13426611 0.70 CD274 (0.48) CYP4F2CYP4A11PIM1MCL1PDE8B
SCHEMBL116636 0.69 CYP2A6 (0.62) PIM1KDM4EALDH1A1SMN1; SMN2CYP2A6
SCHEMBL14688685 0.69 PIM1 (0.41) ATRCYP4F2CYP4A11PIM1CHRNB2
SCHEMBL14688512 0.69 PIM1 (0.41) ATRCYP4F2CYP4A11PIM1MCL1
SCHEMBL14688800 0.69 CYP4F2 (0.40) CYP4F2CYP4A11PIM1MCL1
SCHEMBL18448117 0.68 MCL1 (0.45) CYP4F2CYP4A11MCL1PDE8BTNF
SCHEMBL14688791 0.68 ATR (0.39) ATRCYP4F2CYP4A11CHRNB2CHRNA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2742046-A1 PYRAZOLO[3,4-c]PYRIDINE COMPOUNDS AND METHODS OF USE F.HOFFMANN-LA ROCHE AG (CH) 2014-06-18 EP disclosed
WO-2013024002-A1 PYRAZOLO[3,4-c]PYRIDINE COMPOUNDS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2013-02-21 WO disclosed