SCHEMBL14710706

SCHEMBL14710706

CCc1cc(F)c(Br)cc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 8/20 0.47
KDM1B Q8NB78 5/20 0.47
KCNH2 Q12809 4/20 0.37
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
TSHR P16473 2/20 0.35
LMNA P02545 1/20 0.35
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.31
PARP1 P09874 1/20 0.31
GPR27 Q9NS67 1/20 0.31
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30871762 0.83 KDM1A (0.47) KDM1AKDM1BKCNH2CYP1A2CYP2D6
SCHEMBL14292894 0.82 KDM1A (0.39) KDM1AKDM1BKCNH2GABRA1GABRB2
SCHEMBL13898962 0.81 NOS3 (0.40) NOS3NOS1NOS2TSHRNPSR1
SCHEMBL22664895 0.81 KDM1A (0.50) KDM1AKDM1BKCNH2CYP1A2ALDH1A1
SCHEMBL18784110 0.81 KDM1A (0.46) KDM1AKDM1BKCNH2CYP1A2CYP2D6
SCHEMBL31414094 0.81 KDM1A (0.46) KDM1AKDM1BKCNH2ALDH1A1
SCHEMBL27918435 0.80 KDM1A (0.42) KDM1AKDM1BKCNH2
SCHEMBL17244913 0.79 ALDH1A1 (0.39) NOS3NOS1NOS2TSHRLMNA
SCHEMBL15250021 0.79 NOS3 (0.39) NOS3NOS1NOS2TSHRNPSR1
SCHEMBL23490846 0.79 KDM1A (0.41) KDM1AKDM1BTSHRNPSR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013025733-A1 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS INTERMUNE, INC. (US) 2013-02-21 WO disclosed