SCHEMBL14713166

SCHEMBL14713166

CC#Cc1cncc(C(=O)N=S(C)(=O)c2ccc(Cl)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.44
PDGFRB P09619 10/20 0.44
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
EGFR P00533 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
F10 P00742 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL835541 0.92 KDR (0.47) KDRPDGFRBPTGS1PTGS2EGFR
SCHEMBL14713178 0.89 KDR (0.42) KDRPDGFRBPTGS1PTGS2PTGDR2
SCHEMBL14713129 0.89 KDR (0.53) KDRPDGFRBPTGS2EGFRLMNA
SCHEMBL1478732 0.89 KDR (0.49) KDRPDGFRBPTGS1PTGS2PTGDR2
SCHEMBL833427 0.88 KDR (0.47) KDRPDGFRBPTGS1PTGS2EGFR
SCHEMBL14713208 0.88 KDR (0.46) KDRPDGFRBPTGDR2
SCHEMBL835000 0.88 KDR (0.52) KDRPDGFRBPTGS1PTGS2PTGDR2
SCHEMBL834233 0.88 KDR (0.42) KDRPDGFRBPTGS1PTGS2EGFR
SCHEMBL836423 0.88 KDR (0.52) KDRPDGFRBPTGS1PTGS2PTGDR2
SCHEMBL836783 0.87 KDR (0.45) KDRPDGFRBPTGS1PTGS2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099757-B1 SULFOXIMINES AS KINASE INHIBITORS ALLERGAN INC (US) 2014-06-25 EP disclosed
US-8383825-B2 Kinase inhibitors ALLERGAN, INC. (US) 2013-02-26 US disclosed