SCHEMBL14713862

SCHEMBL14713862

Cc1c2cc(-c3cccnc3)ncc2nn1COCC[Si](C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 13/20 0.46
PIM3 Q86V86 3/20 0.46
PIM2 Q9P1W9 3/20 0.46
CYP2A6 P11509 4/20 0.41
DGAT1 O75907 1/20 0.39
CYP3A4 P08684 2/20 0.37
CYP2E1 P05181 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2B6 P20813 2/20 0.37
CYP2C19 P33261 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14688648 0.90 PIM1 (0.43) PIM1PIM3PIM2CYP2A6DGAT1
SCHEMBL14713858 0.83 CYP2A6 (0.41) PIM1PIM3PIM2CYP2A6DGAT1
SCHEMBL14688761 0.80 DGAT1 (0.40) PIM1PIM3PIM2CYP2A6DGAT1
SCHEMBL14689121 0.79 DGAT1 (0.38) PIM1PIM3PIM2CYP2A6DGAT1
SCHEMBL14688516 0.79 PIM1 (0.49) PIM1PIM3PIM2CYP2A6DGAT1
SCHEMBL14688835 0.77 PIM1 (0.52) PIM1PIM3PIM2CYP2A6DGAT1
SCHEMBL14688870 0.75 PIM1 (0.53) PIM1PIM3PIM2DGAT1MAPT
SCHEMBL14689482 0.75 PIM1 (0.50) PIM1PIM3PIM2DGAT1MAPT
SCHEMBL14689125 0.75 PIM1 (0.41) PIM1PIM3PIM2DGAT1
SCHEMBL14689076 0.75 PIM1 (0.38) PIM1PIM3PIM2CYP2A6DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013024002-A1 PYRAZOLO[3,4-c]PYRIDINE COMPOUNDS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2013-02-21 WO disclosed