SCHEMBL14715434

SCHEMBL14715434

COc1cc2nc(N3CCC(CC4CC4)(OC(=O)N(C)Cc4ccccc4)CC3)nc(O)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EHMT2 Q96KQ7 7/20 0.44
WHR1 P49842 2/20 0.42
DNMT3A Q9Y6K1 1/20 0.42
NSD2 O96028 1/20 0.42
EZH2 Q15910 1/20 0.42
NSD3 Q9BZ95 1/20 0.42
EHMT1 Q9H9B1 1/20 0.42
KIT P10721 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715415 0.97 EHMT2 (0.43) EHMT2WHR1DNMT3ANSD2EZH2
SCHEMBL14715412 0.90 WHR1 (0.44) EHMT2WHR1
SCHEMBL2172163 0.87 EHMT2 (0.45) EHMT2WHR1DNMT3ANSD2EZH2
SCHEMBL14715363 0.85 EHMT2 (0.44) EHMT2WHR1DNMT3ANSD2EZH2
SCHEMBL2174116 0.84 EHMT2 (0.44) EHMT2WHR1DNMT3ANSD2EZH2
SCHEMBL14715357 0.82 EHMT2 (0.45) EHMT2WHR1DNMT3ANSD2EZH2
SCHEMBL2170980 0.80 WHR1 (0.48) EHMT2WHR1
SCHEMBL2172172 0.80 EHMT2 (0.41) EHMT2WHR1DNMT3ANSD2EZH2
SCHEMBL2173189 0.78 EHMT2 (0.46) EHMT2WHR1DNMT3ANSD2EZH2
SCHEMBL2170894 0.78 WHR1 (0.49) WHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed