SCHEMBL14715412

SCHEMBL14715412

COc1cc2nc(N3CCC(Cc4ccccc4)(OC(=O)N(C)Cc4ccccc4)CC3)nc(O)c2cc1OC

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
WHR1 P49842 3/20 0.44
EHMT2 Q96KQ7 1/20 0.43
ADRA1A P35348 3/20 0.42
ADRA1B P35368 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715434 0.90 EHMT2 (0.44) WHR1EHMT2
SCHEMBL14715415 0.89 EHMT2 (0.43) WHR1EHMT2
SCHEMBL2170980 0.86 WHR1 (0.48) WHR1EHMT2ADRA1AADRA1B
SCHEMBL14715376 0.84 WHR1 (0.46) WHR1EHMT2ADRA1AADRA1B
SCHEMBL2170706 0.81 WHR1 (0.51) WHR1EHMT2ADRA1AADRA1B
SCHEMBL14715407 0.81 EHMT2 (0.48) WHR1EHMT2ADRA1AADRA1B
SCHEMBL14715393 0.81 EHMT2 (0.45) WHR1EHMT2ADRA1AADRA1B
SCHEMBL2172163 0.80 EHMT2 (0.45) WHR1EHMT2
SCHEMBL14715448 0.80 ADRA2A (0.47) WHR1EHMT2ADRA1AADRA1B
SCHEMBL13361589 0.80 WHR1 (0.49) WHR1ADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed