SCHEMBL14715455

SCHEMBL14715455

COc1cc2nc(N3CCC(Cc4ccccc4)(OC(=O)NC4Cc5ccccc5C4)CC3)nc(N)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.55
ADRA1B P35368 4/20 0.55
TP53 P04637 1/20 0.49
GLA P06280 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
TSHR P16473 1/20 0.49
ADRA1D P25100 1/20 0.49
THPO P40225 1/20 0.49
HIF1A Q16665 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715170 0.95 ADRA1A (0.51) ADRA1AADRA1BTP53GLACYP3A4
SCHEMBL14715393 0.92 EHMT2 (0.45) ADRA1AADRA1B
SCHEMBL14715365 0.89 ADRA1A (0.49) ADRA1AADRA1BADRA1D
SCHEMBL14715261 0.88 ADRA1A (0.49) ADRA1AADRA1BTP53GLACYP3A4
SCHEMBL3319567 0.87 ADRA1A (0.56) ADRA1AADRA1B
SCHEMBL14715308 0.87 ADRA1A (0.49) ADRA1AADRA1BADRA1D
SCHEMBL14715370 0.87 EHMT2 (0.44) ADRA1AADRA1B
SCHEMBL14715262 0.87 ADRA1A (0.56) ADRA1AADRA1BTP53GLACYP3A4
SCHEMBL14715452 0.86 ADRA1A (0.48) ADRA1AADRA1BADRA1D
SCHEMBL3673034 0.85 ADRA1A (0.54) ADRA1AADRA1BADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed