SCHEMBL3673034

SCHEMBL3673034

COc1cc2nc(N3CCC(Cc4ccccc4)(C(=O)NC4Cc5ccccc5C4)CC3)nc(N)c2cc1OC.COc1cc2nc(N3CCC(Cc4ccccc4)(C(=O)O)CC3)nc(N)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.54
ADRA1B P35368 4/20 0.54
ADRA1D P25100 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3319567 0.98 ADRA1A (0.56) ADRA1AADRA1B
SCHEMBL13333056 0.92 ADRA1A (0.53) ADRA1AADRA1BADRA1D
SCHEMBL3320049 0.90 ADRA1A (0.56) ADRA1AADRA1BADRA1D
SCHEMBL2176843 0.90 EHMT2 (0.46) ADRA1AADRA1B
SCHEMBL2173344 0.89 ADRA1A (0.61) ADRA1AADRA1BADRA1D
SCHEMBL2207053 0.89 ADRA1A (0.48) ADRA1AADRA1BADRA1D
SCHEMBL13333050 0.86 ADRA1A (0.51) ADRA1AADRA1B
SCHEMBL13333054 0.86 ADRA1A (0.50) ADRA1AADRA1B
SCHEMBL14715455 0.85 ADRA1A (0.55) ADRA1AADRA1BADRA1D
SCHEMBL7919688 0.85 EHMT2 (0.45) ADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010054968-A1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-05-20 WO claimed
WO-2010054968-A1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-05-20 WO disclosed