SCHEMBL14715684

SCHEMBL14715684

N#Cc1cc(F)ccc1OC1CCN(CC[C@H]2CC[C@H](NC(=O)OC3CCOCC3)CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 9/20 0.46
HTR2A P28223 8/20 0.46
TBK1 Q9UHD2 8/20 0.43
IKBKE Q14164 5/20 0.43
DRD2 P14416 6/20 0.42
HTR1A P08908 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3083241 0.90 DRD3 (0.57) DRD3HTR2ADRD2
SCHEMBL14715621 0.87 HTR2A (0.47) DRD3HTR2ADRD2HTR1A
SCHEMBL3963444 0.87 DRD2 (0.56) DRD3HTR2ADRD2HTR1A
SCHEMBL3075427 0.87 DRD2 (0.56) DRD3HTR2ADRD2HTR1A
SCHEMBL3067525 0.86 DRD3 (0.53) DRD3HTR2ADRD2
SCHEMBL3078178 0.86 DRD3 (0.53) DRD3HTR2ADRD2
SCHEMBL3091198 0.85 DRD3 (0.47) DRD3HTR2ADRD2HTR1A
SCHEMBL3083297 0.85 DRD3 (0.47) DRD3HTR2ADRD2HTR1A
SCHEMBL3080661 0.85 DRD3 (0.49) DRD3HTR2ADRD2
SCHEMBL14715609 0.85 HRH1 (0.45) DRD3HTR2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed