Vincamine

Vincamine

SCHEMBL147179

CC[C@]12CCCN3CCc4c(n(c5ccccc45)[C@@](O)(C(=O)OC)C1)[C@@H]32

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 1.00
KCNH2 Q12809 3/20 1.00
CYP2D6 P10635 3/20 1.00
HIF1A Q16665 3/20 1.00
MEN1 O00255 3/20 1.00
KMT2A Q03164 3/20 1.00
KDM4E B2RXH2 2/20 1.00
MAPT P10636 2/20 1.00
GAA P10253 1/20 1.00
CASP6 P55212 1/20 1.00
L3MBTL1 Q9Y468 1/20 1.00
NR1I2 O75469 3/20 0.78
PDE4D Q08499 2/20 0.78
HRH3 Q9Y5N1 2/20 0.78
OPRK1 P41145 1/20 0.78
LMNA P02545 3/20 0.57
CYP1A2 P05177 2/20 0.57
TSHR P16473 2/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Vincamine SCHEMBL14095103 1.00 CYP3A4 (1.00) CYP3A4KCNH2CYP2D6HIF1AMEN1
Vincamine SCHEMBL3767 1.00 CYP3A4 (1.00) CYP3A4KCNH2CYP2D6HIF1AMEN1
Vincamine SCHEMBL30892136 1.00 CYP3A4 (1.00) CYP3A4KCNH2CYP2D6HIF1AMEN1
Vincamine SCHEMBL29710919 1.00 CYP3A4 (1.00) CYP3A4KCNH2CYP2D6HIF1AMEN1
Vincamine SCHEMBL8970683 1.00 CYP3A4 (1.00) CYP3A4KCNH2CYP2D6HIF1AMEN1
Vincamine SCHEMBL8134417 0.99 CYP3A4 (0.98) CYP3A4KCNH2CYP2D6HIF1AMEN1
Vincamine SCHEMBL6631357 0.98 CYP3A4 (0.96) CYP3A4KCNH2CYP2D6HIF1AMEN1
Vincamine SCHEMBL5712113 0.98 CYP3A4 (0.96) CYP3A4KCNH2CYP2D6HIF1AMEN1
Vincamine SCHEMBL6162410 0.97 CYP3A4 (0.95) CYP3A4KCNH2CYP2D6HIF1AMEN1
Vincamine SCHEMBL11619815 0.97 CYP3A4 (0.93) CYP3A4KCNH2CYP2D6HIF1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6584 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4739310-A1 ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE 1 (ENPP1) INHIBITOR COMBINATIONS AND USES THEREOF Insilico Medicine IP Limited (HK) 2026-05-13 EP claimed
US-20260035369-A1 VINCAMINE DERIVATIVES, PREPARATION METHOD THEREFOR, AND USE THEREOF UNIV SOUTHWEST (CN) 2026-02-05 US claimed
US-20250339399-A1 SUPRAMOLECULAR SELF-ASSEMBLY SYSTEM BEIJING CREATRON INSTITUTE OF PHARMACEUTICAL RES CO LTD (CN) 2025-11-06 US claimed
EP-4642484-A1 TARGETED TREATMENT OF PROSTATE CANCERS AND OTHER TUMORS BY AN ANTIBODY-DRUG CONJUGATE Hangzhou Seehe Biotechnology Co., Ltd (CN) 2025-11-05 EP claimed
EP-4642492-A1 AN ANTIBODY-DRUG CONJUGATE HAVING TWO OR MORE FUNCTIONAL SMALL MOLECULE COMPOUNDS FOR ENHANCED TREATMENT OF REFRACTORY DISEASES Hangzhou Seehe Biotechnology Co., Ltd (CN) 2025-11-05 EP claimed
US-20250313900-A1 COMPOSITIONS AND THERAPEUTIC AGENTS FOR MODULATING INFLAMMATORY RESPONSES ON BOTH TUMOR AND IMMUNE CELLS THE METHODIST HOSPITAL 2025-10-09 US claimed
US-12419860-B2 Time release sleep aid system NIGHTWISE, LLC (US) 2025-09-23 US claimed
CN-116731010-B Vincamine derivative, and preparation method and application thereof 西南大学 2025-02-11 CN claimed
WO-2025007955-A1 ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE 1 (ENPP1) INHIBITOR COMBINATIONS AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2025-01-09 WO claimed
US-20240415810-A1 TIME RELEASE SLEEP AID SYSTEM NIGHTWISE, LLC 2024-12-19 US claimed
EP-0007823-A2 3,20-Dioxo-4,9-diene-21-hydroxy-steroid compounds, process for their preparation, their use in medicines and pharmaceutical compositions containing them ROUSSEL-UCLAF (FR) 1980-02-06 EP claimed
EP-0005100-A1 Epoxidation reagent and its use for the epoxidation of acyclic, cyclic or polycyclic organic compounds containing at least one ethylenic unsaturation ROUSSEL-UCLAF (FR) 1979-10-31 EP claimed
EP-0004222-A1 4,5-Seco-estrane-3,5,17-trione derivatives, process for their preparation and their use for the preparation of therapeutically active compounds ROUSSEL-UCLAF (FR) 1979-09-19 EP claimed
US-4140777-A Cerebral vasodilating 6-substituted vincamines ENRICO CORVI MORA (IT) 1979-02-20 US claimed
US-4122179-A VASODILATORS Mora, Enrico Corvi (IT) 1978-10-24 US claimed
US-4021559-A 6,7-DIHYDROXYCOUMARIN-4-METHYL-SULFONIC ACID SYNTHELABO (FR) 1977-05-03 US claimed
US-3979395-A Process for the preparation of vincamine and other indole alkaloids BUSKINE S.A. (CH) 1976-09-07 US claimed
US-3957981-A CEREBRAL VASODILATORS PARCOR (FR) 1976-05-18 US claimed
US-3957995-A ADMINISTERING, CEREBRAL VASODILATOR ACTIVITY PARCOR (FR) 1976-05-18 US claimed
US-3937709-A ENAMINES, ALKYLATION, METHYL A-BROMOMETHYL ACRYLATE, REDUCTION, OXIDATION, CYCLIZATION AGENCE NATIONALE DE VALORISATION DE LA RECHERCHE (ANVAR) (FR) 1976-02-10 US claimed