SCHEMBL14720542

SCHEMBL14720542

Brc1ccc(C=C2CCN(CC3CC3)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 8/20 0.56
THRB P10828 1/20 0.40
CCR2 P41597 1/20 0.40
IKBKB O14920 1/20 0.39
KCNH2 Q12809 1/20 0.39
HTR7 P34969 1/20 0.38
MAOB P27338 1/20 0.37
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
SIGMAR1 Q99720 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20333309 0.84 MCHR1 (0.46) MCHR1CCR2MAOBHTR2AHTR2C
SCHEMBL20305006 0.80 SRD5A2 (0.54) MCHR1HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL14721386 0.79 GPR183 (0.49) MCHR1
SCHEMBL20304836 0.76 MCHR1 (0.54) MCHR1THRB
SCHEMBL14720870 0.76 MCHR1 (0.52) MCHR1HTR7HTR2AHTR2C
SCHEMBL14721932 0.74 GPR183 (0.45) MCHR1
SCHEMBL14720920 0.73 HRH3 (0.47) MCHR1KCNH2HTR7
SCHEMBL14720608 0.73 HRH3 (0.43) MCHR1KCNH2MAOB
SCHEMBL12891140 0.73 MAOA (0.45) MAOB
SCHEMBL14720741 0.71 OPRM1 (0.44) MCHR1HTR2CSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed