SCHEMBL14723649

SCHEMBL14723649

CC(C)(C)OC(=O)Nc1ccc(Oc2ccnc(N)c2OCc2ccccc2)c2cccnc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 1/20 0.45
HDAC1 Q13547 2/20 0.39
CYP2C9 P11712 1/20 0.37
PTGER1 P34995 1/20 0.37
MAPK14 Q16539 2/20 0.37
LTA4H P09960 1/20 0.37
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KDM4E B2RXH2 1/20 0.36
RPS6KB1 P23443 2/20 0.35
BRAF P15056 1/20 0.35
AURKA O14965 1/20 0.35
METAP1 P53582 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
AAK1 Q2M2I8 1/20 0.35
TLR7 Q9NYK1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14723651 0.87 SLC40A1 (0.41) SLC40A1CYP2C9PTGER1ALDH1A1SMN1; SMN2
SCHEMBL12790198 0.84 HTT (0.41) MAPK14ALDH1A1SMN1; SMN2HPGDHTT
SCHEMBL13667124 0.84 METAP1 (0.41) MAPK14ALDH1A1SMN1; SMN2HPGDHTT
SCHEMBL13667088 0.80 KDM4E (0.39) HDAC1CYP2C9ALDH1A1SMN1; SMN2HPGD
SCHEMBL12847501 0.80 MAPT (0.39) ALDH1A1SMN1; SMN2HPGDHTTHSD17B10
SCHEMBL12847422 0.77 SRC (0.41) MAPK14KDM4EBRAFAURKAMETAP1
SCHEMBL2936138 0.76 BRAF (0.43) MAPK14BRAFAURKAAAK1SRC
SCHEMBL13666962 0.74 MAPT (0.35) ALDH1A1SMN1; SMN2HPGDHTTHSD17B10
SCHEMBL6279532 0.73 BRD4 (0.48) SLC40A1HDAC1CYP2C9PTGER1MEN1
SCHEMBL12847306 0.73 MAPT (0.43) MAPK14KDM4EBRAFMETAP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8383816-B2 Aryl-quinolyl compounds and their use CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2013-02-26 US disclosed