SCHEMBL14724286

SCHEMBL14724286

Bc1cnc(-c2cccc(Cc3nnc4ccc(C(=O)OCCCC)nn34)c2)nc1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MET P08581 17/20 0.38
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12224224 0.92 MET (0.38) METPDE3BPDE3AKDM4EALDH1A1
SCHEMBL2528823 0.92 MET (0.38) METPDE3BPDE3AKDM4EALDH1A1
SCHEMBL14724340 0.89 MET (0.42) MET
SCHEMBL12224264 0.80 MET (0.43) MET
SCHEMBL12224223 0.80 MET (0.43) METKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL2529553 0.79 MET (0.42) MET
SCHEMBL14724301 0.79 MET (0.44) MET
SCHEMBL14715581 0.78 MET (0.35) METMAPT
SCHEMBL12224263 0.78 MET (0.43) METKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL12224222 0.76 MET (0.42) MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367827-B1 3-(3-PYRIMIDINE-2-YL-BENZYL)-[1,2,4]TRIAZOLO [4,3-b]PYRIDAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2013-02-27 EP disclosed