SCHEMBL14730465

SCHEMBL14730465

N#Cc1cc(NC=O)ccc1F

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.48
EGLN2 Q96KS0 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
BLM P54132 1/20 0.40
WRN Q14191 1/20 0.40
PGR P06401 1/20 0.39
ALDH1A1 P00352 1/20 0.38
PTP4A3 O75365 1/20 0.38
TRPV4 Q9HBA0 2/20 0.37
AR P10275 2/20 0.37
SLC22A12 Q96S37 1/20 0.35
CNR2 P34972 1/20 0.35
ACLY P53396 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19144095 0.85 EGLN2 (0.50) EGLN2PGRALDH1A1TRPV4
SCHEMBL8410428 0.82 ALDH1A1 (0.44) EGLN2ABCG2ALDH1A1SLC22A12
SCHEMBL546977 0.79 SLC22A12 (0.56) ARSLC22A12CNR2
SCHEMBL3173181 0.79 GRM4 (0.48) GRM4ABCG2BLMWRNPGR
SCHEMBL241795 0.78 RAB9A (0.46) ALDH1A1SLC22A12
SCHEMBL8410032 0.78 SLC22A12 (0.51) GRM4BLMWRNALDH1A1TRPV4
SCHEMBL21844923 0.77 GRM4 (0.47) GRM4ABCG2BLMWRNPGR
SCHEMBL19190440 0.77 GRM4 (0.50) GRM4ABCG2BLMWRNPGR
SCHEMBL897882 0.77 GRM4 (0.47) GRM4ABCG2BLMWRNPGR
SCHEMBL7230699 0.76 GRM4 (0.46) GRM4ABCG2BLMWRNPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3712139-A1 ANTI-HBV TETRAHYDROISOXAZOLO[4,3-C]PYRIDINE COMPOUNDS Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2020-09-23 EP disclosed
WO-2019154343-A1 CAPSID PROTEIN ASSEMBLY INHIBITOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 正大天晴药业集团股份有限公司 2019-08-15 WO disclosed
WO-2013027196-A1 SUBSTITUTED 2-ALKYL-1-OXO-N-PHENYL-3-HETEROARYL-1,2,3,4- TETRAHYDROISOQUINOLINE-4-CARBOXAMIDES FOR ANTIMALARIAL THERAPIES ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2013-02-28 WO disclosed