SCHEMBL14733012

SCHEMBL14733012

Cc1nc(-c2cccc(CCCc3cccc(-c4nc(C)c5ccccc5n4)n3)n2)nc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.47
CYP1A2 P05177 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
NUDT1 P36639 1/20 0.42
HSD17B10 Q99714 1/20 0.42
GPR3 P46089 1/20 0.42
TGFBR1 P36897 5/20 0.40
MAPK14 Q16539 1/20 0.40
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
RAB9A P51151 2/20 0.38
MPO P05164 1/20 0.37
RAD52 P43351 1/20 0.37
METAP1 P53582 1/20 0.37
KCNH2 Q12809 1/20 0.37
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14732922 0.93 TGFBR1 (0.47) PDE10ACYP1A2ALDH1A1HPGDNUDT1
SCHEMBL8779392 0.84 PDE10A (0.46) PDE10ACYP1A2ALDH1A1HPGDNUDT1
SCHEMBL14733019 0.80 METAP1 (0.49) TGFBR1MAPK14KMT2AMEN1RAB9A
SCHEMBL14733018 0.80 TGFBR1 (0.46) TGFBR1MAPK14NOS3NOS1NOS2
SCHEMBL8779715 0.79 MAPT (0.44) PDE10ACYP1A2ALDH1A1HPGDNUDT1
SCHEMBL8884919 0.78 PDE10A (0.62) PDE10ACYP1A2ALDH1A1HPGDNUDT1
SCHEMBL8779730 0.77 PDE10A (0.40) PDE10ACYP1A2ALDH1A1HPGDNUDT1
SCHEMBL8872433 0.76 PDE10A (0.49) PDE10ACYP1A2ALDH1A1HPGDNUDT1
SCHEMBL14732960 0.73 CYP1A2 (0.42) PDE10ACYP1A2GPR3KCNH2L3MBTL1
SCHEMBL8779683 0.71 GRM5 (0.53) PDE10ACYP1A2ALDH1A1HPGDNUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026866-A2 NOVEL MICROBIOCIDES SYNGENTA PARTICIPATIONS AG (CH) 2013-02-28 WO disclosed