SCHEMBL14743302

SCHEMBL14743302

COc1ccc(CN(C(=O)c2ccccc2)c2cc(C(=O)O)cc3cc(Cl)cc(Cl)c23)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
BCL2A1 Q16548 2/20 0.45
PDK1 Q15118 1/20 0.45
LPAR1 Q92633 2/20 0.44
LPAR5 Q9H1C0 2/20 0.44
TAS2R14 Q9NYV8 4/20 0.43
PTGES O14684 2/20 0.42
ALOX5 P09917 1/20 0.42
STAT3 P40763 1/20 0.42
TSHR P16473 2/20 0.42
TAS2R8 Q9NYW2 1/20 0.41
CXCR3 P49682 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEP1A Q16819 1/20 0.41
MEP1B Q16820 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14743329 0.92 NPC1 (0.45) NPC1RAB9AMEN1KMT2ABCL2A1
SCHEMBL14743730 0.90 PTGES (0.55) NPC1RAB9AMEN1KMT2ALPAR1
SCHEMBL14743655 0.90 TSHR (0.42) NPC1MEN1KMT2APDK1PTGES
SCHEMBL14743067 0.85 ALDH1A1 (0.43) NPC1RAB9AMEN1KMT2APDK1
SCHEMBL14743568 0.83 MRGPRX4 (0.36) NPC1RAB9AMEN1KMT2APTGES
SCHEMBL14743539 0.83 PTGES (0.48) NPC1RAB9ALPAR1LPAR5TAS2R14
SCHEMBL14743558 0.82 ALDH1A1 (0.45) MEN1KMT2ATSHR
SCHEMBL14743729 0.80 PTGES (0.47) MEN1KMT2ATAS2R14PTGESALOX5
SCHEMBL14743619 0.80 ALDH1A1 (0.38) MEN1KMT2ATDP1
SCHEMBL14743090 0.80 MEN1 (0.43) RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013030358-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2013-03-07 WO disclosed