SCHEMBL14743449

SCHEMBL14743449

O=C(C[S+]([O-])c1cccc(Cl)c1)Nc1ccc(C(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNJ5 P48544 1/20 0.48
KCNJ3 P48549 1/20 0.48
P2RX4 Q99571 2/20 0.45
P2RX1 P51575 1/20 0.45
P2RX7 Q99572 1/20 0.45
TMPRSS4 Q9NRS4 1/20 0.45
RHOC P08134 6/20 0.45
RHOA P61586 6/20 0.45
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
GRIK1 P39086 1/20 0.43
BAZ1A Q9NRL2 1/20 0.42
MTOR P42345 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
EPHX2 P34913 1/20 0.42
NLRP3 Q96P20 1/20 0.42
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14743066 0.86 KMT2A (0.47) P2RX1ALDH1A1MEN1KMT2A
SCHEMBL14744258 0.86 KMT2A (0.47) P2RX1ALDH1A1MEN1KMT2A
SCHEMBL14743338 0.86 KMT2A (0.47) P2RX1ALDH1A1MEN1KMT2A
SCHEMBL14743056 0.85 KMT2A (0.49) ALDH1A1HPGDL3MBTL1EPHX2NLRP3
SCHEMBL14743396 0.81 ADORA3 (0.51) ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL14743511 0.81 MAPT (0.47) TMPRSS4ALDH1A1NLRP3MEN1POLB
SCHEMBL14743584 0.81 ADORA3 (0.51) ALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL14743391 0.81 MEN1 (0.57) KCNJ5KCNJ3ALDH1A1HPGDGRIK1
SCHEMBL29475999 0.77 GRIN2B (0.43) ALDH1A1MEN1KMT2A
SCHEMBL14743029 0.76 GRIK1 (0.44) ALDH1A1GRIK1L3MBTL1MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2758370-A1 PARP INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2014-07-30 EP claimed
WO-2013030205-A1 PARP INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2013-03-07 WO claimed
EP-2758370-A1 PARP INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2014-07-30 EP disclosed
WO-2013030205-A1 PARP INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2013-03-07 WO disclosed