SCHEMBL14744109

SCHEMBL14744109

COC(=O)[C@H]1COC(CCNC(=O)OC(C)(C)C)=N1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 3/20 0.39
GFER P55789 1/20 0.39
EPHX1 P07099 1/20 0.38
TDP1 Q9NUW8 2/20 0.38
MAN2B1 O00754 1/20 0.38
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPT P10636 1/20 0.36
LMNA P02545 1/20 0.35
NQO2 P16083 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14737595 1.00 HTT (0.43) HTTNPSR1ALDH1A1GFEREPHX1
SCHEMBL3583570 0.87 L3MBTL1 (0.39) HTTNPSR1GFEREPHX1MAN2B1
SCHEMBL28230784 0.83 HTT (0.45) HTTNPSR1ALDH1A1GFEREPHX1
SCHEMBL12299216 0.79 MEN1 (0.39) HTTNPSR1ALDH1A1GFEREPHX1
SCHEMBL18764623 0.78 HTT (0.43) HTTNPSR1ALDH1A1GFEREPHX1
SCHEMBL18764829 0.78 HTT (0.45) HTTNPSR1ALDH1A1GFEREPHX1
SCHEMBL30322973 0.75 PEPD (0.35) LMNA
SCHEMBL28231758 0.74 HTT (0.46) HTTNPSR1ALDH1A1GFEREPHX1
SCHEMBL18792409 0.73 MIF (0.31)
SCHEMBL30562984 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763990-A1 PYRROLOPYRAZINE KINASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2014-08-13 EP disclosed
WO-2013030138-A1 PYRROLOPYRAZINE KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2013-03-07 WO disclosed