SCHEMBL14744157

SCHEMBL14744157

N#Cc1ccccc1-c1c(Cl)cc(N)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.42
ESR2 Q92731 1/20 0.41
AR P10275 1/20 0.39
ALDH1A1 P00352 6/20 0.38
KDM4E B2RXH2 4/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
USP8 P40818 1/20 0.37
USP7 Q93009 1/20 0.37
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
HPGD P15428 3/20 0.36
MAPT P10636 2/20 0.36
GRIA1 P42261 1/20 0.36
CACNG8 Q8WXS5 1/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 1/20 0.36
GALR3 O60755 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14744345 0.78 RORC (0.45) RORCARALDH1A1KDM4EADORA2A
SCHEMBL17266575 0.72 LRRK2 (0.49) ESR2ARALDH1A1KDM4EADORA2A
SCHEMBL27909137 0.72 ESR2 (0.52) ESR2ALDH1A1KDM4EUSP8USP7
SCHEMBL3259923 0.72 CYP1A2 (0.47) ESR2ALDH1A1KDM4EADORA2AUSP8
SCHEMBL14744241 0.72 PLA2G7 (0.55) ALDH1A1KDM4EGABRG2GABRB3GABRA5
SCHEMBL16013714 0.72 CYP3A4 (0.39) ALDH1A1KDM4EADORA2AADORA1CYP3A4
SCHEMBL38650555 0.72 CYP1A1 (0.42) ALDH1A1ADORA2AHPGDMAPTPOLB
SCHEMBL22664353 0.71 RORC (0.36) RORCARALDH1A1KDM4EHPGD
SCHEMBL222 0.71 ESR2 (0.60) ESR2ARALDH1A1KDM4EUSP8
SCHEMBL29412287 0.71 ESR2 (0.60) ESR2ARALDH1A1KDM4EUSP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed