SCHEMBL14747749

SCHEMBL14747749

COCCCN1C(=O)C(C)Oc2cc(CI)c(C)cc21

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
REN P00797 5/20 0.47
TSHR P16473 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP3A4 P08684 3/20 0.39
CYP2C19 P33261 3/20 0.39
ALDH1A1 P00352 4/20 0.36
THRB P10828 1/20 0.36
CYP1A2 P05177 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2C9 P11712 1/20 0.35
PPARG P37231 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7636421 0.89 REN (0.53) RENTSHRNPSR1CYP3A4CYP2C19
SCHEMBL14747751 0.87 REN (0.42) RENTSHRNPSR1ALDH1A1THRB
SCHEMBL5987076 0.86 REN (0.49) RENTSHRNPSR1CYP3A4CYP2C19
SCHEMBL5986192 0.84 REN (0.48) RENTSHRNPSR1CYP3A4CYP2C19
SCHEMBL7634836 0.84 REN (0.48) RENTSHRNPSR1CYP3A4CYP2C19
SCHEMBL5985048 0.84 REN (0.48) RENTSHRNPSR1CYP3A4CYP2C19
SCHEMBL14747753 0.81 CYP2C19 (0.42) RENTSHRNPSR1CYP3A4CYP2C19
SCHEMBL5985698 0.81 REN (0.46) RENTSHRNPSR1CYP3A4CYP2C19
SCHEMBL5987063 0.81 REN (0.46) RENTSHRNPSR1CYP3A4CYP2C19
SCHEMBL13434135 0.79 TSHR (0.59) RENTSHRNPSR1CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8389511-B2 Bicyclic heterocyclic derivative DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2013-03-05 US disclosed