SCHEMBL14747801

SCHEMBL14747801

OCc1ccc(-c2cc(C(F)(F)F)nn2-c2ccccc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 5/20 0.74
PTGS2 P35354 10/20 0.70
CYP2C9 P11712 1/20 0.61
PDPK1 O15530 3/20 0.61
MAPT P10636 2/20 0.56
TP53 P04637 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27602808 0.86 PTGS1 (0.74) PTGS1PTGS2CYP2C9PDPK1
SCHEMBL27339504 0.86 PTGS1 (0.68) PTGS1PTGS2CYP2C9PDPK1MAPT
SCHEMBL6451398 0.85 PTGS1 (1.00) PTGS1PTGS2PDPK1MAPTTP53
SCHEMBL6097735 0.84 PTGS1 (0.70) PTGS1PTGS2CYP2C9PDPK1
SCHEMBL27602805 0.83 PTGS1 (0.82) PTGS1PTGS2PDPK1MAPTTP53
SCHEMBL9089381 0.83 PTGS2 (0.79) PTGS1PTGS2CYP2C9PDPK1
Primary Alcohol Metabolite Of Celecoxib SCHEMBL6013984 0.83 PTGS2 (1.00) PTGS1PTGS2CYP2C9PDPK1
SCHEMBL6757697 0.83 PTGS2 (0.79) PTGS1PTGS2CYP2C9PDPK1
Carbamic Acid SCHEMBL5860891 0.83 PTGS2 (0.69) PTGS1PTGS2CYP2C9PDPK1MAPT
SCHEMBL5344449 0.82 PTGS1 (0.80) PTGS1PTGS2CYP2C9PDPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44048-E1 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-YL]benzenesulfonamide for the treatment of inflammation or an inflammation-associated disorder G.D. SEARLE LLC (US) 2013-03-05 US disclosed