SCHEMBL5344449

SCHEMBL5344449

Cc1ccc(-c2cc(C(F)(F)F)nn2-c2ccccc2)cc1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 7/20 0.80
PTGS2 P35354 10/20 0.70
CYP2C9 P11712 3/20 0.70
PDPK1 O15530 3/20 0.68
HDAC3 O15379 2/20 0.68
HDAC4 P56524 2/20 0.68
HDAC1 Q13547 2/20 0.68
HDAC7 Q8WUI4 2/20 0.68
HDAC2 Q92769 2/20 0.68
HDAC10 Q969S8 2/20 0.68
HDAC11 Q96DB2 2/20 0.68
HDAC8 Q9BY41 2/20 0.68
HDAC6 Q9UBN7 2/20 0.68
HDAC9 Q9UKV0 2/20 0.68
HDAC5 Q9UQL6 2/20 0.68
ALOX5 P09917 2/20 0.68
PTGES O14684 1/20 0.68
CA12 O43570 1/20 0.68
PDE5A O76074 1/20 0.68
ABCB11 O95342 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14198881 0.94 PTGS1 (0.80) PTGS1PTGS2CYP2C9PDPK1HDAC3
SCHEMBL8266070 0.92 PTGS2 (0.80) PTGS1PTGS2CYP2C9PDPK1HDAC3
Carbamic Acid SCHEMBL5859288 0.92 PTGS1 (0.68) PTGS1PTGS2CYP2C9PDPK1HDAC3
Sulfamide SCHEMBL7136410 0.92 PTGS2 (0.78) PTGS1PTGS2CYP2C9PDPK1HDAC3
SCHEMBL15915380 0.92 PTGS1 (0.68) PTGS1PTGS2CYP2C9PDPK1HDAC3
SCHEMBL6451398 0.89 PTGS1 (1.00) PTGS1PTGS2PDPK1MAPTSMN1; SMN2
SCHEMBL5426104 0.89 PTGS2 (0.63) PTGS1PTGS2CYP2C9PDPK1HDAC3
SCHEMBL4587051 0.87 PTGS2 (0.73) PTGS1PTGS2CYP2C9PDPK1HDAC3
SCHEMBL8265772 0.87 PTGS2 (0.73) PTGS1PTGS2CYP2C9PDPK1HDAC3
SCHEMBL27602805 0.87 PTGS1 (0.82) PTGS1PTGS2PDPK1MAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111499576-A Preparation method of celecoxib impurity 迪嘉药业集团有限公司 2020-08-07 CN claimed
EP-0731795-A1 SUBSTITUTED PYRAZOLYL BENZENESULFONAMIDES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP claimed
EP-2445343-B1 PRODRUGS OF NH-ACIDIC COMPOUNDS ALKERMES PHARMA IRELAND LTD (IE) 2021-08-04 EP disclosed
CN-111499576-A Preparation method of celecoxib impurity 迪嘉药业集团有限公司 2020-08-07 CN disclosed
CN-111499576-A Preparation method of celecoxib impurity 迪嘉药业集团有限公司 2020-08-07 CN disclosed
US-7202367-B2 Process for arylating or vinylating or alkynating a nucleophilic compound RHODIA CHIMIE (FR) 2007-04-10 US disclosed
US-7202367-B2 Process for arylating or vinylating or alkynating a nucleophilic compound RHODIA CHIMIE (FR) 2007-04-10 US disclosed
US-20070060629-A1 Large conductance calcium-activated k channel opener TANABE SEIYAKU CO., LTD. (JP) 2007-03-15 US disclosed
US-20070060629-A1 Large conductance calcium-activated k channel opener TANABE SEIYAKU CO., LTD. (JP) 2007-03-15 US disclosed
US-20070060629-A1 Large conductance calcium-activated k channel opener TANABE SEIYAKU CO., LTD. (JP) 2007-03-15 US disclosed
EP-1675585-A2 LARGE CONDUCTANCE CALCIUM-ACTIVATED K CHANNEL OPENER TANABE SEIYAKU CO., LTD. (JP) 2006-07-05 EP disclosed
US-20050234239-A1 Method of forming a carbon-carbon or carbon-heteroatom linkage SHASUN PHARMA SOLUTIONS, INC. 2005-10-20 US disclosed
CN-1668595-A Method for forming carbon-carbon or carbon-heteroatom bonds RHONE POULENC CHIMIE (FR) 2005-09-14 CN disclosed
EP-1562914-A1 NITRIC OXIDE RELEASING SELECTIVE CYCLOOXYGENASE-2 INHIBITORS Merck Frosst Canada & Co. (CA) 2005-08-17 EP disclosed
WO-2005037271-A2 LARGE CONDUCTANCE CALCIUM-ACTIVATED K CHANNEL OPENER TANABE SEIYAKU CO., LTD. (JP) 2005-04-28 WO disclosed
EP-1509502-A1 METHOD OF FORMING A CARBON-CARBON OR CARBON-HETEROATOM LINKAGE RHODIA CHIMIE (FR) 2005-03-02 EP disclosed
WO-2004037798-A1 NITRIC OXIDE RELEASING SELECTIVE CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA & CO. (CA) 2004-05-06 WO disclosed
US-20030236413-A1 Catalysis in presence of a metallic element, an imine ligand and nitrogen compound as chelating compound, forming a chemical intermediates in the agrochemical and pharmaceutical fields SHASUN PHARMA SOLUTIONS, INC. 2003-12-25 US disclosed
WO-2003101966-A1 METHOD OF FORMING A CARBON-CARBON OR CARBON-HETEROATOM LINKAGE RHODIA CHIMIE (FR) 2003-12-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050234239-A1 Method of forming a carbon-carbon or carbon-heteroatom linkage AOC1, AOC3, NUDT1 PTGS1 1096/4885PTGS2 965/4885CYP2C9 258/4885
US-20030236413-A1 Catalysis in presence of a metallic element, an imine ligand and nitrogen compound as chelating compound, forming a chemical intermediates in the agrochemical and pharmaceutical fields ALK, INMT, ACHE PTGS1 2593/4885PTGS2 2246/4885CYP2C9 24/4885
US-20070060629-A1 Large conductance calcium-activated k channel opener KCNN3, KCNN1, KCNN2 PTGS1 558/4885PTGS2 594/4885CYP2C9 1249/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.