SCHEMBL14748448

SCHEMBL14748448

N#Cc1ccc(Oc2ccc3c(c2)COB3)cc1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 9/20 0.41
PDE4A P27815 4/20 0.37
PDE4C Q08493 4/20 0.37
PDE4D Q08499 4/20 0.37
CHRM1 P11229 1/20 0.37
ADRA1A P35348 1/20 0.37
PDE1A P54750 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE7A Q13946 1/20 0.37
PDE3A Q14432 1/20 0.37
POLB P06746 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.34
PRKAB2 O43741 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA2 P54646 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAG3 Q9UGI9 1/20 0.33
PRKAG2 Q9UGJ0 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14748450 0.83 PDE4B (0.44) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL7997145 0.80 AR (0.45) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL14470676 0.78 PDE4B (0.53) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL14748456 0.77 CTNNB1 (0.42) POLB
SCHEMBL19622210 0.76 PDE4B (0.44) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL2527560 0.75 PDE4B (0.74) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL8004927 0.75 PDE4B (0.56) PDE4BPDE4APDE4CPDE4DPOLB
SCHEMBL14748463 0.75 PDE4B (0.47) PDE4BPDE4APDE4CPDE4DPOLB
SCHEMBL8007244 0.75 PDE4B (0.42) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL5801556 0.74 PDE4A (0.49) PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed
EP-2564857-B1 Boron-containing small molecules as anti-inflammatory agents ANACOR PHARMACEUTICALS INC (US) 2017-05-03 EP disclosed
EP-2564857-A1 Boron-containing small molecules as anti-inflammatory agents Anacor Pharmaceuticals, Inc. (US) 2013-03-06 EP disclosed